SCHEMBL9307979

SCHEMBL9307979

CCc1ccc2c(C)cc(=O)[nH]c2c1

nearest known ligand 0.59

Predicted protein targets (top 17)

geneUniProtsupporting neighboursconfidence
KDM4E B2RXH2 5/20 0.59
GLA P06280 3/20 0.59
GAA P10253 3/20 0.59
ALDH1A1 P00352 3/20 0.59
HPGD P15428 2/20 0.59
TP53 P04637 1/20 0.59
SMN1; SMN2 Q16637 1/20 0.59
TNKS2 Q9H2K2 8/20 0.55
CYP1A2 P05177 1/20 0.55
CYP2C19 P33261 1/20 0.55
KIF11 P52732 1/20 0.54
TNKS O95271 1/20 0.48
LMNA P02545 1/20 0.46
PPARA Q07869 1/20 0.45
DAO P14920 1/20 0.45
HSD17B10 Q99714 1/20 0.44
MAPT P10636 1/20 0.44

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL2056350 0.86 LMNA (0.59) KDM4EGLAGAAALDH1A1HPGD
SCHEMBL15828752 0.84 KDM4E (0.62) KDM4EGLAGAAALDH1A1HPGD
SCHEMBL13267221 0.83 KDM4E (0.54) KDM4EGLAGAAALDH1A1HPGD
SCHEMBL278605 0.78 KIF11 (0.81) KDM4EALDH1A1CYP1A2KIF11DAO
SCHEMBL29864765 0.78 KIF11 (0.81) KDM4EALDH1A1CYP1A2KIF11DAO
SCHEMBL19032120 0.77 LMNA (0.60) KDM4EGAAALDH1A1HPGDSMN1; SMN2
SCHEMBL2795205 0.77 KDM4E (0.67) KDM4EGLAGAAALDH1A1HPGD
SCHEMBL13560650 0.76 KIF11 (0.61) KDM4EGLAGAAALDH1A1HPGD
SCHEMBL7028425 0.75 KIF11 (0.54) KDM4EGAAALDH1A1HPGDTP53
SCHEMBL22501754 0.75 AR (0.69) KDM4EGLAGAAALDH1A1HPGD

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5371226-A Hypotensive agents MERCK PATENT GESELLSCHAFT MIT BESCHRANKTER HAFTUNG (DE) 1994-12-06 US disclosed
CN-1077192-A The 2-oxoquinoline derivatives MERCK PATENT GMBH (DE) 1993-10-13 CN disclosed
EP-0561252-A1 2-Oxoquinoline derivatives as angiotensin II antagonists MERCK PATENT GmbH (DE) 1993-09-22 EP disclosed