SCHEMBL9309739

SCHEMBL9309739

CCc1nc(C)nc(NN)c1Cc1ccc(-c2ccccc2C#N)cc1

nearest known ligand 0.40

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
PPARG P37231 2/20 0.39
GRM5 P41594 1/20 0.37
ALDH1A1 P00352 4/20 0.36
CYP1A2 P05177 3/20 0.36
CYP3A4 P08684 3/20 0.36
HSD17B10 Q99714 3/20 0.36
MAPK1 P28482 2/20 0.36
CLK4 Q9HAZ1 2/20 0.36
ESR2 Q92731 1/20 0.36
CYP2C9 P11712 2/20 0.35
TSHR P16473 2/20 0.35
KDM4E B2RXH2 2/20 0.35
HPGD P15428 2/20 0.35
TP53 P04637 1/20 0.35
MYC P01106 1/20 0.35
WDR5 P61964 1/20 0.35
MEN1 O00255 2/20 0.34
KMT2A Q03164 2/20 0.34
USP2 O75604 1/20 0.34
CYP2D6 P10635 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9308565 0.92 PPARG (0.45) PPARG
SCHEMBL9308911 0.90 PPARG (0.41) PPARGALDH1A1KDM4EHPGDACHE
SCHEMBL9309571 0.84 ESR2 (0.45) PPARGESR2MYCWDR5GRIA2
SCHEMBL9309094 0.82 PPARG (0.36) PPARGALDH1A1CYP1A2CYP3A4HSD17B10
SCHEMBL9308516 0.82 PPARG (0.44) PPARGALDH1A1CYP1A2CYP3A4HSD17B10
SCHEMBL9308512 0.81 PPARG (0.45) PPARGALDH1A1CYP1A2CYP3A4HSD17B10
SCHEMBL9308652 0.81 PPARG (0.43) PPARGALDH1A1CYP1A2CYP3A4HSD17B10
SCHEMBL9308631 0.80 CYP19A1 (0.41) PPARGGRM5ALDH1A1CYP1A2CYP2C9
SCHEMBL9308992 0.78 CYP1A2 (0.45) PPARGALDH1A1CYP1A2CYP3A4HSD17B10
SCHEMBL1895309 0.76 KDM4E (0.41) PPARGALDH1A1CYP1A2MAPK1ESR2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5358950-A Useful in treatment of cardiovascular diseases LABORATOIRES UPSA (FR) 1994-10-25 US disclosed