SCHEMBL9318010

SCHEMBL9318010

O=C(O)CCN1CC(=O)N(c2ccccc2)c2ccc(I)cc2C1=O

nearest known ligand 0.50

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
KDM4E B2RXH2 3/20 0.50
ALOX15 P16050 1/20 0.50
TSHR P16473 1/20 0.50
SIRT1 Q96EB6 1/20 0.50
ITGB3 P05106 2/20 0.44
ITGA2B P08514 2/20 0.44
ENPP2 Q13822 2/20 0.38
MDM2 Q00987 4/20 0.38
MEN1 O00255 2/20 0.37
KMT2A Q03164 2/20 0.37
POLB P06746 1/20 0.37
MAPT P10636 1/20 0.37
TDP1 Q9NUW8 1/20 0.37
L3MBTL1 Q9Y468 1/20 0.37
OPRK1 P41145 1/20 0.36
PDE4D Q08499 1/20 0.36
ALDH1A1 P00352 2/20 0.36
HPGD P15428 2/20 0.36
CES2 O00748 1/20 0.36
BCHE P06276 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9318151 0.90 MDM2 (0.46) KDM4EALOX15TSHRSIRT1ITGB3
SCHEMBL9319073 0.87 MDM2 (0.41) KDM4EALOX15TSHRSIRT1ITGB3
SCHEMBL7332495 0.87 ALDH1A1 (0.40) KDM4EALOX15TSHRSIRT1ITGB3
SCHEMBL8959460 0.81 KDM4E (0.47) KDM4EALOX15TSHRSIRT1ITGB3
SCHEMBL7322450 0.79 KDM4E (0.43) KDM4EALOX15TSHRSIRT1ITGB3
SCHEMBL7326762 0.77 AGTR1 (0.39) KDM4ETSHRMDM2POLBMAPT
SCHEMBL7329007 0.76 ALDH1A1 (0.37) KDM4EMEN1KMT2APOLBMAPT
SCHEMBL7332551 0.74 PPARD (0.41) ALOX15MDM2MEN1KMT2AALDH1A1
Trifluoroacetic Acid SCHEMBL7333942 0.73 ITGB3 (0.70) KDM4EALOX15TSHRSIRT1ITGB3
SCHEMBL7329841 0.72 ITGB3 (0.44) KDM4EALOX15TSHRSIRT1ITGB3

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0610334-A1 NONPEPTIDYL INTEGRIN INHIBITORS HAVING SPECIFICITY FOR THE GPII b?III a? RECEPTOR. GENENTECH INC (US) 1994-08-17 EP disclosed