SCHEMBL9318151

SCHEMBL9318151

O=C(O)CCN1CC(=O)N(c2ccc(Cl)cc2)c2ccc(I)cc2C1=O

nearest known ligand 0.46

Predicted protein targets (top 9)

geneUniProtsupporting neighboursconfidence
MDM2 Q00987 16/20 0.46
ITGB3 P05106 1/20 0.42
ITGA2B P08514 1/20 0.42
TP53 P04637 1/20 0.42
KDM4E B2RXH2 1/20 0.42
ALOX15 P16050 1/20 0.42
TSHR P16473 1/20 0.42
SIRT1 Q96EB6 1/20 0.42
AGTR1 P30556 1/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9318010 0.90 KDM4E (0.50) MDM2ITGB3ITGA2BKDM4EALOX15
SCHEMBL9319073 0.87 MDM2 (0.41) MDM2ITGB3ITGA2BTP53KDM4E
SCHEMBL7326762 0.86 AGTR1 (0.39) MDM2TP53KDM4ETSHRAGTR1
SCHEMBL7332495 0.78 ALDH1A1 (0.40) ITGB3ITGA2BKDM4EALOX15TSHR
Trifluoroacetic Acid SCHEMBL7331122 0.77 ITGB3 (0.37) MDM2ITGB3ITGA2BKDM4EALOX15
Trifluoroacetic Acid SCHEMBL7333020 0.77 ITGB3 (0.37) MDM2ITGB3ITGA2BKDM4EALOX15
SCHEMBL7329007 0.75 ALDH1A1 (0.37) KDM4E
SCHEMBL8959460 0.74 KDM4E (0.47) MDM2ITGB3ITGA2BTP53KDM4E
SCHEMBL11692626 0.74 KMT2A (0.50) KDM4EALOX15TSHRSIRT1
SCHEMBL7332551 0.74 PPARD (0.41) MDM2ALOX15

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0610334-A1 NONPEPTIDYL INTEGRIN INHIBITORS HAVING SPECIFICITY FOR THE GPII b?III a? RECEPTOR. GENENTECH INC (US) 1994-08-17 EP disclosed