SCHEMBL9318596

SCHEMBL9318596

c1ccc(C[N+]2CCCC2)cc1

nearest known ligand 0.42

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
TP53 P04637 1/20 0.42
CHKA P35790 4/20 0.41
CALM1 P0DP23 1/20 0.39
ALDH1A1 P00352 5/20 0.36
LMNA P02545 3/20 0.36
HTT P42858 2/20 0.36
SMN1; SMN2 Q16637 2/20 0.36
TSHR P16473 3/20 0.36
IDO1 P14902 1/20 0.36
LOXL2 Q9Y4K0 1/20 0.36
TRPA1 O75762 1/20 0.36
KDM4E B2RXH2 1/20 0.36
TDP1 Q9NUW8 1/20 0.36
SIGMAR1 Q99720 1/20 0.36
SLC6A3 Q01959 1/20 0.35
MAOB P27338 1/20 0.35
HPGD P15428 1/20 0.35
ALOX15 P16050 1/20 0.35
ALOX12 P18054 1/20 0.35
CASP1 P29466 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL368538 0.98 CHKA (0.40) TP53CHKACALM1ALDH1A1LMNA
SCHEMBL6549159 0.90 TP53 (0.46) TP53CHKACALM1ALDH1A1LMNA
SCHEMBL5100518 0.81 TP53 (0.39) TP53CHKACALM1ALDH1A1LMNA
SCHEMBL11155177 0.79 SIGMAR1 (0.44) TP53CALM1ALDH1A1TSHRSIGMAR1
SCHEMBL27609076 0.76 ACHE (0.47) TP53ALDH1A1HTTSIGMAR1
SCHEMBL348590 0.76 ALDH1A1 (0.39) TP53ALDH1A1TSHR
SCHEMBL349052 0.73 GBA1 (0.39) ALDH1A1SMN1; SMN2TSHRTDP1
SCHEMBL7283642 0.72 CHKA (0.36) TP53CHKACALM1ALDH1A1LMNA
SCHEMBL368873 0.71 ESR2 (0.38) TSHRKDM4ETDP1SIGMAR1HSD17B10
SCHEMBL11347488 0.71 SLC18A3 (0.47) ALDH1A1LMNAHTTTSHRSIGMAR1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5051432-A Heterocyclic 1,4 dihydropyridine derivatives GLAXO, S.P.A. (IT) 1991-09-24 US claimed
EP-0238211-B1 Dihydropyridines, process for their preparation and their use as medicaments GLAXO SPA (IT) 1994-01-12 EP disclosed
US-5051432-A Heterocyclic 1,4 dihydropyridine derivatives GLAXO, S.P.A. (IT) 1991-09-24 US disclosed
EP-0238211-A2 Dihydropyridines, process for their preparation and their use as medicaments GLAXO S.p.A. (IT) 1987-09-23 EP disclosed