SCHEMBL9318772

SCHEMBL9318772

CNC(=O)c1c(I)cc(I)c(C(N)=O)c1I

nearest known ligand 0.36

Predicted protein targets (top 17)

geneUniProtsupporting neighboursconfidence
TP53 P04637 1/20 0.36
PLAU P00749 1/20 0.34
MKNK2 Q9HBH9 1/20 0.33
NEU3 Q9UQ49 1/20 0.33
IKBKB O14920 1/20 0.32
TSHR P16473 1/20 0.32
MAPK1 P28482 1/20 0.32
CHEK1 O14757 1/20 0.31
MAP4K4 O95819 1/20 0.31
EGFR P00533 1/20 0.31
HDAC8 Q9BY41 2/20 0.31
HDAC6 Q9UBN7 2/20 0.31
BRD4 O60885 1/20 0.31
HDAC2 Q92769 1/20 0.31
CREBBP Q92793 1/20 0.30
CA2 P00918 1/20 0.30
POLB P06746 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL3932936 0.84 TPMT (0.37) TSHRMAPK1POLB
SCHEMBL7158495 0.83 TSHR (0.46) TP53NEU3TSHRMAPK1CHEK1
SCHEMBL11297490 0.82 POLB (0.34) TP53PLAUMKNK2NEU3TSHR
SCHEMBL3663229 0.76 TSHR (0.46) TSHRMAPK1POLB
SCHEMBL3398797 0.76 HPGD (0.37) CHEK1CA2POLB
SCHEMBL9787517 0.76 LMNA (0.35) NEU3BRD4POLB
SCHEMBL8359643 0.75 LMNA (0.47) TSHRMAPK1POLB
SCHEMBL9787542 0.75 HDAC8 (0.37) TP53TSHREGFRHDAC8HDAC6
SCHEMBL9451092 0.75 POLB (0.32) TSHRMAPK1POLB
SCHEMBL29423654 0.75 POLB (0.32) TSHRMAPK1POLB

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0558484-A1 NOVEL X-RAY CONTRAST AGENTS, COMPOSITIONS AND METHODS MALLINCKRODT MEDICAL, INC. (US) 1993-09-08 EP claimed
WO-1992009562-A1 NOVEL X-RAY CONTRAST AGENTS, COMPOSITIONS AND METHODS MALLINCKRODT MEDICAL, INC. (US) 1992-06-11 WO claimed
US-5356613-A X-ray contrast agents, compositions and methods MALLINCKRODT MEDICAL, INC. (US) 1994-10-18 US disclosed