SCHEMBL9326801

SCHEMBL9326801

CCCCCCCCCCCCC(NC(=O)C(F)(F)F)c1coc([Si](C)(C)C)c1

nearest known ligand 0.37

Predicted protein targets (top 12)

geneUniProtsupporting neighboursconfidence
EPHX1 P07099 1/20 0.37
MLYCD O95822 3/20 0.36
TACR3 P29371 2/20 0.36
ASAH1 Q13510 1/20 0.32
ALDH1A1 P00352 1/20 0.31
FAAH O00519 7/20 0.31
CES1 P23141 5/20 0.31
CES2 O00748 2/20 0.31
MEN1 O00255 1/20 0.31
CYP1A2 P05177 1/20 0.31
KMT2A Q03164 1/20 0.31
HSD17B10 Q99714 1/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9325177 0.85 ALDH1A1 (0.39) TACR3ALDH1A1
SCHEMBL9744772 0.83 TACR3 (0.37) EPHX1TACR3FAAH
SCHEMBL9328354 0.83 TACR3 (0.37) TACR3
SCHEMBL9767101 0.78 FAAH (0.37) ALDH1A1FAAHCES1CES2MEN1
SCHEMBL7326578 0.77 ALDH1A1 (0.38) TACR3ALDH1A1
SCHEMBL9326410 0.76 CA2 (0.32)
SCHEMBL7303995 0.74 CA2 (0.40) ALDH1A1MEN1CYP1A2KMT2A
SCHEMBL7301168 0.74 CA2 (0.40) ALDH1A1MEN1CYP1A2KMT2A
SCHEMBL9671527 0.74 CA2 (0.40) ALDH1A1MEN1CYP1A2KMT2A
SCHEMBL9671129 0.74 CA2 (0.40) ALDH1A1MEN1CYP1A2KMT2A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 6 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5322953-A Antiinflammatory agents; intermediates for 2-furanone compounds ALLERGAN, INC. (US) 1994-06-21 US disclosed
US-5298633-A Silane intermediates ALLERGAN, INC. (US) 1994-03-29 US disclosed
US-5171863-A 2-trialkylsily-4-substituted furan derivatives ALLERGAN, INC. (US) 1992-12-15 US disclosed
US-5089485-A ANTI-INFLAMMATORY FURANONES ALLERGAN, INC. (US) 1992-02-18 US disclosed
US-5082954-A Intermediates and processes for preparing 4-substituted 2-5(H)-furanones as anti-inflammatory agents ALLERGAN, INC. (US) 1992-01-21 US disclosed
EP-0369811-A2 Anti-inflammatory furanones ALLERGAN, INC (US) 1990-05-23 EP disclosed