SCHEMBL9329501

SCHEMBL9329501

O=[C]CC(=O)c1cccs1

nearest known ligand 0.64

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 3/20 0.64
NPC1 O15118 2/20 0.64
RAB9A P51151 2/20 0.64
LMNA P02545 2/20 0.64
MEN1 O00255 2/20 0.64
POLB P06746 2/20 0.64
KMT2A Q03164 2/20 0.64
GSK3B P49841 1/20 0.60
HPGD P15428 5/20 0.55
SMN1; SMN2 Q16637 1/20 0.55
ERCC5 P28715 1/20 0.55
FEN1 P39748 1/20 0.55
CES2 O00748 1/20 0.54
CES1 P23141 1/20 0.54
DAO P14920 1/20 0.52
TSHR P16473 2/20 0.51
PKM P14618 1/20 0.51
MAPK1 P28482 1/20 0.51
HTT P42858 1/20 0.51
HSD17B10 Q99714 1/20 0.51

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL137872 0.82 ALDH1A1 (0.62) ALDH1A1NPC1RAB9ALMNAMEN1
SCHEMBL711360 0.79 RAB9A (0.75) ALDH1A1NPC1RAB9ALMNAMEN1
SCHEMBL2216212 0.79 ALDH1A1 (1.00) ALDH1A1NPC1RAB9ALMNAMEN1
SCHEMBL23855456 0.77
SCHEMBL8505274 0.76 ALDH1A1 (0.58) ALDH1A1NPC1RAB9ALMNAMEN1
SCHEMBL658097 0.75
SCHEMBL11407883 0.75
SCHEMBL230036 0.75
SCHEMBL22721189 0.75 ALDH1A1 (0.83) ALDH1A1NPC1RAB9ALMNAMEN1
SCHEMBL9608874 0.75

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 12 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0225634-B1 Antibacterial compounds, their production and use TAKEDA CHEMICAL INDUSTRIES LTD (JP) 1994-04-06 EP disclosed
US-4946837-A ANTIBIOTICS TAKEDA CHEMICAL INDUSTRIES, LTD. (JP) 1990-08-07 US disclosed
US-4839351-A Antibacterial compounds, and use TAKEDA CHEMICAL INDUSTRIES, LTD. (JP) 1989-06-13 US disclosed
US-4826834-A BACTERICIDES TAKEDA CHEMICAL INDUSTRIES, LTD. (JP) 1989-05-02 US disclosed
US-4788185-A Cephalosporin compounds TAKEDA CHEMICAL INDUSTRIES, LTD. (JP) 1988-11-29 US disclosed
EP-0229369-A2 Cephalosporins, process for their preparation and pharmaceutical compositions containing them Takeda Chemical Industries, Ltd. (JP) 1987-07-22 EP disclosed
EP-0225634-A2 Antibacterial compounds, their production and use Takeda Chemical Industries, Ltd. (JP) 1987-06-16 EP disclosed
US-4665065-A 3-pyrazolo(1,5-aαpyridinium cephem compounds TAKEDA CHEMICAL INDUSTRIES, LTD. (JP) 1987-05-12 US disclosed
EP-0216385-A2 Antibacterial compounds Takeda Chemical Industries, Ltd. (JP) 1987-04-01 EP disclosed
EP-0164113-A2 3-pyrazolo(1,5-a)pyridinium cephem compounds, their production and use Takeda Chemical Industries, Ltd. (JP) 1985-12-11 EP disclosed
EP-0164122-A2 Cephem compounds Takeda Chemical Industries, Ltd. (JP) 1985-12-11 EP disclosed
EP-0160252-A2 Antibacterial compounds Takeda Chemical Industries, Ltd. (JP) 1985-11-06 EP disclosed