SCHEMBL9330232

SCHEMBL9330232

CCCOC([O])(c1nnnn1-c1ccncc1)c1nnnn1C(C)c1ccccc1

nearest known ligand 0.40

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 9/20 0.40
ROCK2 O75116 2/20 0.37
HTT P42858 2/20 0.36
MAPT P10636 1/20 0.36
HPGD P15428 1/20 0.36
CCR6 P51684 1/20 0.36
CACNA1B Q00975 1/20 0.36
APBA1 Q02410 1/20 0.36
NPSR1 Q6W5P4 2/20 0.34
MEN1 O00255 2/20 0.33
KMT2A Q03164 2/20 0.33
TP53 P04637 1/20 0.33
ATM Q13315 1/20 0.33
TSHR P16473 1/20 0.33
PKM P14618 1/20 0.31
CYP1A2 P05177 2/20 0.31
CYP3A4 P08684 2/20 0.31
GABRA1 P14867 2/20 0.31
GABRB2 P47870 2/20 0.31
CYP11B1 P15538 2/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9755577 0.85 ALDH1A1 (0.36) ALDH1A1ROCK2HTTMAPTHPGD
SCHEMBL9755580 0.71 PKM (0.32) ALDH1A1HTTKMT2APKMLMNA
SCHEMBL25669632 0.67 NPSR1 (0.39) ALDH1A1ROCK2HTTMAPTHPGD
SCHEMBL9330238 0.67 HSD11B1 (0.36) ALDH1A1ROCK2HTTNPSR1MEN1
SCHEMBL9329826 0.66 ALDH1A1 (0.53) ALDH1A1HTTMAPTHPGDCCR6
SCHEMBL7317875 0.66 FAAH (0.36) ALDH1A1ROCK2HTTMAPTNPSR1
SCHEMBL8881199 0.61 DAGLA (0.39) ALDH1A1ROCK2HTTMAPTHPGD
SCHEMBL96013 0.61 FAAH (0.39) ALDH1A1ROCK2HTTMAPTHPGD
SCHEMBL22952393 0.60 ALDH1A1 (0.57) ALDH1A1HTTMAPTHPGDCCR6
SCHEMBL24038267 0.60 MEN1 (0.46) ROCK2HPGDNPSR1MEN1KMT2A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5302613-A Antiatheroscleroic and antithrombotic 2-amino-6-phenyl-4H-pyran-4-ones THE UPJOHN COMPANY (US) 1994-04-12 US disclosed
US-5252735-A Antiatherosclerotic and antithrombotic 2-amino-6-phenyl-4H-pyran-4-ones THE UPJOHN COMPANY (US) 1993-10-12 US disclosed