SCHEMBL933898

SCHEMBL933898

CC(Cc1ccc(-c2ccncc2)cc1)C(N)=O

nearest known ligand 0.49

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CYP17A1 P05093 2/20 0.49
CYP3A4 P08684 2/20 0.46
ALDH1A1 P00352 1/20 0.46
AAK1 Q2M2I8 1/20 0.44
MMP12 P39900 1/20 0.44
MMP13 P45452 1/20 0.44
LRRK2 Q5S007 4/20 0.44
EPHX1 P07099 1/20 0.44
ROCK2 O75116 4/20 0.43
ROCK1 Q13464 4/20 0.43
PRKACA P17612 2/20 0.43
IRAK1 P51617 2/20 0.43
PRKX P51817 2/20 0.43
PRKG1 Q13976 2/20 0.43
PKN2 Q16513 2/20 0.43
CLK4 Q9HAZ1 2/20 0.43
RPS6KB1 P23443 1/20 0.43
LIMK1 P53667 1/20 0.43
PRKG2 Q13237 1/20 0.43
HIPK4 Q8NE63 1/20 0.43

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL1286079 0.90 CYP3A4 (0.54) CYP17A1CYP3A4ALDH1A1EPHX1TBXAS1
SCHEMBL933922 0.83 MKNK1 (0.55) MMP12LRRK2TBXAS1F10PRSS1
SCHEMBL933472 0.83 PRKCI (0.54) CYP3A4ALDH1A1LRRK2ROCK2ROCK1
SCHEMBL26167691 0.83 SRR (0.54)
SCHEMBL5027971 0.81 CYP17A1 (0.50) CYP17A1CYP3A4AAK1MMP12MMP13
SCHEMBL934557 0.77 EPHX1 (0.39) EPHX1TBXAS1
SCHEMBL23643108 0.77 EPHX1 (0.50) EPHX1F10
SCHEMBL934530 0.77 TAAR1 (0.59) EPHX1
SCHEMBL22593510 0.77 EPHX1 (0.50) EPHX1MAPK1
SCHEMBL22937469 0.77 EPHX1 (0.50) CYP3A4ALDH1A1EPHX1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2011006935-A2 TETRAZOLE DERIVATIVES MERCK SERONO S.A. (CH) 2011-01-20 WO disclosed