SCHEMBL9339092

SCHEMBL9339092

O=C(CCC1CCN(C(=O)OCc2ccccc2)CC1)Nc1cccc(C(=O)NCCC(=O)OCc2ccccc2)c1

nearest known ligand 0.46

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
HTT P42858 1/20 0.46
CYP2C9 P11712 3/20 0.46
CYP3A4 P08684 2/20 0.46
KMT2A Q03164 2/20 0.46
SMN1; SMN2 Q16637 2/20 0.46
MEN1 O00255 1/20 0.46
ALDH1A1 P00352 1/20 0.46
CYP1A2 P05177 1/20 0.46
MAPT P10636 1/20 0.46
CYP2C19 P33261 1/20 0.46
GRIN2B Q13224 3/20 0.45
CYP2D6 P10635 2/20 0.45
RAB9A P51151 2/20 0.44
NPC1 O15118 1/20 0.44
CCKBR P32239 1/20 0.43
KDM4E B2RXH2 1/20 0.43
FAAH O00519 1/20 0.43
F13A1 P00488 1/20 0.43
TGM2 P21980 1/20 0.43
TGM1 P22735 1/20 0.43

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL10444861 0.94 ITGB3 (0.46) HTTCYP2C9CYP3A4KMT2ASMN1; SMN2
SCHEMBL7900109 0.85 MAPT (0.49) HTTCYP2C9CYP3A4KMT2ASMN1; SMN2
SCHEMBL7909493 0.84 F13A1 (0.44) HTTKMT2ASMN1; SMN2MEN1ALDH1A1
SCHEMBL8381979 0.81 MAPT (0.48) SMN1; SMN2MAPTRAB9ANPC1KDM4E
SCHEMBL7909711 0.80 ST14 (0.40) HTTCYP3A4KMT2ASMN1; SMN2MEN1
SCHEMBL9866050 0.80 GAA (0.54) HTTKMT2ASMN1; SMN2MEN1ALDH1A1
SCHEMBL9335780 0.79 ITGB3 (0.50) CYP2C9CYP3A4KMT2ASMN1; SMN2MEN1
SCHEMBL7906634 0.79 MEN1 (0.49) KMT2AMEN1MAPTRAB9AKDM4E
SCHEMBL9865134 0.77 HTT (0.53) HTTKMT2ASMN1; SMN2MEN1ALDH1A1
SCHEMBL8385674 0.77 GLA (0.52) HTTCYP2C9CYP3A4KMT2ASMN1; SMN2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0372486-B1 Benzoic-acid phenylacetic-acid derivatives, their preparation and their use as medicines HOFFMANN LA ROCHE (CH) 1994-06-01 EP disclosed
US-5039805-A Novel benzoic and phenylacetic acid derivatives HOFFMANN-LA ROCHE INC. (US) 1991-08-13 US disclosed