SCHEMBL934419

SCHEMBL934419

N#Cc1cc(N)cc(Cl)c1

nearest known ligand 0.55

Predicted protein targets (top 19)

geneUniProtsupporting neighboursconfidence
CYP3A4 P08684 3/20 0.55
TP53 P04637 1/20 0.55
GRM5 P41594 5/20 0.37
VCAM1 P19320 1/20 0.36
ALDH1A1 P00352 2/20 0.36
EGLN2 Q96KS0 1/20 0.36
MAOA P21397 1/20 0.34
MAOB P27338 1/20 0.34
ADRA1D P25100 1/20 0.34
CYP1A2 P05177 2/20 0.33
MEN1 O00255 2/20 0.33
KMT2A Q03164 2/20 0.33
TTR P02766 1/20 0.33
ALB P02768 1/20 0.33
KDM4E B2RXH2 1/20 0.33
CYP2D6 P10635 1/20 0.33
MAPT P10636 1/20 0.33
HPGD P15428 1/20 0.33
CYP2C19 P33261 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL30407999 1.00 CYP3A4 (0.55) CYP3A4TP53GRM5VCAM1ALDH1A1
SCHEMBL2011602 0.82 TTR (0.40) CYP3A4VCAM1ALDH1A1EGLN2MEN1
SCHEMBL5852713 0.82 VCAM1 (0.43) GRM5VCAM1MAOAMAOBCYP1A2
SCHEMBL3182180 0.82 TTR (0.40) VCAM1ALDH1A1EGLN2MEN1KMT2A
SCHEMBL633226 0.82 TSHR (0.50) CYP3A4TP53GRM5VCAM1MAOA
Hydrochloric Acid SCHEMBL9495207 0.79 TTR (0.39) CYP3A4VCAM1ALDH1A1EGLN2MEN1
SCHEMBL8486211 0.76 CYP3A4 (0.55) CYP3A4TP53ALDH1A1
Water SCHEMBL27778570 0.74 TTR (0.37) VCAM1EGLN2MEN1KMT2ATTR
Nitrogen SCHEMBL28728934 0.73 CYP3A4 (0.87) CYP3A4TP53ALDH1A1
SCHEMBL127074 0.73

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 120 patents — showing the first 20. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-20250340508-A1 TETRAHYDRO-1H-CYCLOPENTA[CD]INDENE DERIVATIVES AS HYPOXIA INDUCIBLE FACTOR-2(ALPHA) INHIBITORS NIKANG THERAPEUTICS INC (US) 2025-11-06 US disclosed
US-12391663-B2 Isoindolinone compounds MONTE ROSA THERAPEUTICS AG (CH) 2025-08-19 US disclosed
US-12391642-B2 Tetrahydro-1H-cyclopenta[cd]indene derivatives as hypoxia inducible factor-2(alpha) inhibitors NIKANG THERAPEUTICS, INC. (US) 2025-08-19 US disclosed
US-12371429-B2 Antibiotic resistance-modifying tricyclic heteroaryl compounds and uses thereof RECREO PHARMACEUTICALS LLC (US) 2025-07-29 US disclosed
US-20240308976-A1 COMPOUNDS THAT MEDIATE PROTEIN DEGRADATION AND USES THEREOF MONTE ROSA THERAPEUTICS AG (CH) 2024-09-19 US disclosed
US-12077506-B2 Indane derivatives as hypoxia inducible factor-2(α) inhibitors NIKANG THERAPEUTICS, INC. (US) 2024-09-03 US disclosed
US-20240261274-A1 TREATMENT OF MYC-DRIVEN CANCERS WITH GSPT1 DEGRADERS MONTE ROSA THERAPEUTICS AG (CH) 2024-08-08 US disclosed
CN-115232026-B Cyano diamine-containing cyano functionalized polyimide mixed matrix membrane and preparation thereof 东华大学 2024-07-30 CN disclosed
US-20240083869-A1 ISOINDOLINONE COMPOUNDS MONTE ROSA THERAPEUTICS AG (CH) 2024-03-14 US disclosed
US-11912682-B2 Isoindolinone compounds MONTE ROSA THERAPEUTICS, INC. (US) 2024-02-27 US disclosed
US-7273882-B2 Aminoacetamide acyl guanidines as β-secretase inhibitors BRISTOL-MYERS SQUIBB COMPANY (US) 2007-09-25 US disclosed
US-7273882-B2 Aminoacetamide acyl guanidines as β-secretase inhibitors BRISTOL-MYERS SQUIBB COMPANY (US) 2007-09-25 US disclosed
US-20070015754-A1 Acyl guanidines as beta-secretase inhibitors BRISTOL-MYERS SQUIBB COMPANY 2007-01-18 US disclosed
US-20070015754-A1 Acyl guanidines as beta-secretase inhibitors BRISTOL-MYERS SQUIBB COMPANY 2007-01-18 US disclosed
US-20070015754-A1 Acyl guanidines as beta-secretase inhibitors BRISTOL-MYERS SQUIBB COMPANY 2007-01-18 US disclosed
WO-2007002214-A2 ACYL GUANIDINES AS BETA-SECRETASE INHIBITORS BRISTOL-MYERS SQUIBB COMPANY (US) 2007-01-04 WO disclosed
WO-2007002214-A2 ACYL GUANIDINES AS BETA-SECRETASE INHIBITORS BRISTOL-MYERS SQUIBB COMPANY (US) 2007-01-04 WO disclosed
WO-2007002220-A2 AMINOACETAMIDE ACYL GUANIDINES AS BETA-SECRETASE INHIBITORS BRISTOL-MYERS SQUIBB COMPANY (US) 2007-01-04 WO disclosed
WO-2007002220-A2 AMINOACETAMIDE ACYL GUANIDINES AS BETA-SECRETASE INHIBITORS BRISTOL-MYERS SQUIBB COMPANY (US) 2007-01-04 WO disclosed
US-20060287287-A1 Aminoacetamide acyl guanidines as beta-secretase inhibitors BRISTOL-MYERS SQUIBB COMPANY 2006-12-21 US disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (11 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-12371429-B2 Antibiotic resistance-modifying tricyclic heteroaryl compounds and uses thereof CBR3, CBR1, CYP2B6 CYP3A4 555/4885TP53 3944/4885GRM5 2852/4885
US-12391663-B2 Isoindolinone compounds CYP4F2, AOC2, AOC3 CYP3A4 684/4885TP53 2966/4885GRM5 3849/4885
US-12077506-B2 Indane derivatives as hypoxia inducible factor-2(α) inhibitors HIF1AN, HIF1A, NFE2L2 CYP3A4 3309/4885TP53 497/4885GRM5 3805/4885
US-20240083869-A1 ISOINDOLINONE COMPOUNDS CYP4F2, AOC2, AOC3 CYP3A4 684/4885TP53 2966/4885GRM5 3849/4885
US-20250340508-A1 TETRAHYDRO-1H-CYCLOPENTA[CD]INDENE DERIVATIVES AS HYPOXIA INDUCIBLE FACTOR-2(ALPHA) INHIBITORS HIF1AN, HIF1A, HYOU1 CYP3A4 2135/4885TP53 1046/4885GRM5 3768/4885
US-12391642-B2 Tetrahydro-1H-cyclopenta[cd]indene derivatives as hypoxia inducible factor-2(alpha) inhibitors HIF1AN, HIF1A, HYOU1 CYP3A4 2135/4885TP53 1046/4885GRM5 3768/4885
US-20060287287-A1 Aminoacetamide acyl guanidines as beta-secretase inhibitors APP, BACE1, BACE2 CYP3A4 3184/4885TP53 1957/4885GRM5 222/4885
US-20240308976-A1 COMPOUNDS THAT MEDIATE PROTEIN DEGRADATION AND USES THEREOF CRBN, GSPT1, GSPT2 CYP3A4 4646/4885TP53 196/4885GRM5 1030/4885
US-11912682-B2 Isoindolinone compounds CYP4F2, AOC2, AOC3 CYP3A4 684/4885TP53 2966/4885GRM5 3849/4885
US-20070015754-A1 Acyl guanidines as beta-secretase inhibitors BACE1, APP, BACE2 CYP3A4 3082/4885TP53 4050/4885GRM5 389/4885
US-20240261274-A1 TREATMENT OF MYC-DRIVEN CANCERS WITH GSPT1 DEGRADERS MYC, MYCBP, GSPT1 CYP3A4 4304/4885TP53 7/4885GRM5 3400/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.