SCHEMBL9347486

SCHEMBL9347486

CCc1cc2c(ccc(=O)n2Cc2ccc(-c3ccccc3-c3nnnn3-c3ccc([N+](=O)[O-])cc3)cc2)c(CC)n1

nearest known ligand 0.43

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
PKM P14618 1/20 0.43
SMN1; SMN2 Q16637 1/20 0.43
PTGS2 P35354 2/20 0.40
AR P10275 1/20 0.39
KMT2A Q03164 2/20 0.38
MEN1 O00255 1/20 0.38
ALOX15 P16050 2/20 0.37
ALOX5 P09917 1/20 0.37
L3MBTL1 Q9Y468 1/20 0.37
AGTR1 P30556 1/20 0.37
P2RX4 Q99571 1/20 0.36
TP53 P04637 1/20 0.36
CYP3A4 P08684 1/20 0.35
CYP2D6 P10635 1/20 0.35
CYP2C9 P11712 1/20 0.35
TSHR P16473 1/20 0.35
MAPK1 P28482 1/20 0.35
CYP2C19 P33261 1/20 0.35
HSD17B10 Q99714 1/20 0.35
CFTR P13569 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9346871 0.83 KMT2A (0.49) SMN1; SMN2KMT2AMEN1L3MBTL1P2RX4
SCHEMBL7276924 0.79 CYP3A4 (0.60) PKMSMN1; SMN2PTGS2ALOX15AGTR1
SCHEMBL9495156 0.77 AGTR1 (0.56) PKMSMN1; SMN2PTGS2KMT2AMEN1
SCHEMBL9494031 0.76 AGTR1 (0.59) PKMSMN1; SMN2PTGS2KMT2AMEN1
SCHEMBL7284844 0.76 AGTR1 (0.43) ALOX15AGTR1CYP3A4CYP2D6CYP2C9
SCHEMBL9312688 0.75 AGTR1 (0.57) AGTR1
Hydrochloric Acid SCHEMBL9350439 0.75 AGTR1 (0.44) ALOX15AGTR1CYP3A4CYP2D6CYP2C9
SCHEMBL9495149 0.74 SMN1; SMN2 (0.45) PKMSMN1; SMN2PTGS2KMT2AAGTR1
SCHEMBL9139431 0.74 AGTR1 (0.54) PKMSMN1; SMN2AGTR1
SCHEMBL7274709 0.73 PPARG (0.52) AGTR1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5294620-A Hypotensive agents or compounds for cardiovascular disorders IMPERIAL CHEMICAL INDUSTRIES PLC (GB) 1994-03-15 US disclosed
US-5217976-A Hypotensive agents, congestive heart failure IMPERIAL CHEMICAL INDUSTRIES PLC (GB) 1993-06-08 US disclosed