SCHEMBL9348336

SCHEMBL9348336

Cc1cc(Cl)ccc1OC#N

nearest known ligand 0.46

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
TSHR P16473 2/20 0.45
HTR2A P28223 1/20 0.45
HTR2C P28335 1/20 0.45
HTR2B P41595 1/20 0.45
MEN1 O00255 4/20 0.44
KMT2A Q03164 4/20 0.44
MAPT P10636 1/20 0.44
SLC6A2 P23975 3/20 0.44
SLC6A4 P31645 3/20 0.44
SLC6A3 Q01959 1/20 0.44
CYP1A2 P05177 2/20 0.42
CYP3A4 P08684 1/20 0.42
CYP2C19 P33261 1/20 0.42
KDM4E B2RXH2 2/20 0.42
ALDH1A1 P00352 2/20 0.42
HPGD P15428 2/20 0.42
SCN4A P35499 2/20 0.41
CYP2C9 P11712 1/20 0.40
HIF1A Q16665 1/20 0.40
TP53 P04637 1/20 0.40

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL10720954 0.90 ESR2 (0.42) TSHRHTR2AHTR2CHTR2BMEN1
SCHEMBL11084242 0.80 TSHR (0.49) TSHRHTR2AHTR2CHTR2BMEN1
SCHEMBL8985167 0.79 GAA (0.44) TSHRMEN1KMT2AMAPTCYP3A4
SCHEMBL11033634 0.79 ALDH1A1 (0.38) TSHRMEN1KMT2AMAPTCYP1A2
SCHEMBL29489134 0.79 GAA (0.44) TSHRMEN1KMT2AMAPTCYP3A4
SCHEMBL9351955 0.79 SLC6A3 (0.47) TSHRMAPTSLC6A2SLC6A4SLC6A3
SCHEMBL9348273 0.78 SLC6A4 (0.48) MEN1KMT2ASLC6A2SLC6A4SLC6A3
SCHEMBL11338994 0.78 AR (0.34) HTR2AMAPTSLC6A4GAA
SCHEMBL807773 0.76 SLC6A2 (0.59) TSHRHTR2AHTR2CHTR2BMEN1
SCHEMBL9419423 0.76 ALDH1A1 (0.39) TSHRMEN1KMT2AKDM4EALDH1A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 7 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0271833-B1 Process for the preparation of aminopyrimidines HOECHST SCHERING AGREVO GMBH (DE) 1994-09-07 EP disclosed
EP-0245901-B1 THIAZINONE DERIVATIVES SHELL INTERNATIONALE RESEARCHMAATSCHAPPIJ B.V. (NL) 1992-08-26 EP disclosed
US-4839356-A FUNGICIDES FOR PLANTS SHELL INTERNATIONALE RESEARCH MAATSCHAPPIJ B.V. (NL) 1989-06-13 US disclosed
US-4833137-A FUNGICIDES FOR PLANTS SHELL INTERNATIONALE RESEARCH MAATSCHAPPIJ B.V. (NL) 1989-05-23 US disclosed
US-4831138-A FROM PROPANEDIIMIDATES DERIVATIVES AND CYANURATES HOECHST AKTIENGESELLSCHAFT (DE) 1989-05-16 US disclosed
EP-0271833-A2 Process for the preparation of aminopyrimidines Hoechst Schering AgrEvo GmbH (DE) 1988-06-22 EP disclosed
EP-0245901-A2 Thiazinone derivatives SHELL INTERNATIONALE RESEARCHMAATSCHAPPIJ B.V. (NL) 1987-11-19 EP disclosed