SCHEMBL9348378

SCHEMBL9348378

CCN(CCc1ccncc1)C(=O)OC(C)(C)C

nearest known ligand 0.44

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
NAMPT P43490 1/20 0.44
CYP17A1 P05093 1/20 0.41
USP2 O75604 1/20 0.40
SSTR4 P31391 1/20 0.39
DAGLB Q8NCG7 2/20 0.39
DAGLA Q9Y4D2 2/20 0.39
LMNA P02545 3/20 0.38
CYP2C9 P11712 3/20 0.38
CYP2C19 P33261 3/20 0.38
CYP1A2 P05177 2/20 0.38
CYP3A4 P08684 2/20 0.38
MEN1 O00255 2/20 0.38
KMT2A Q03164 2/20 0.38
CHRM2 P08172 1/20 0.38
CHRM4 P08173 1/20 0.38
CHRM5 P08912 1/20 0.38
MAPT P10636 1/20 0.38
CHRM1 P11229 1/20 0.38
CHRM3 P20309 1/20 0.38
BLM P54132 1/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL968701 0.85 USP2 (0.51) CYP17A1USP2LMNACYP2C9CYP2C19
SCHEMBL4781274 0.85 HDAC3 (0.48) LMNACYP1A2MEN1KMT2ACHRM2
SCHEMBL31403206 0.84 TRPM8 (0.40) NAMPTMEN1KMT2AHCRTR2HDAC3
SCHEMBL7337070 0.82 CYP17A1 (0.43) CYP17A1CYP2C9CYP2C19CYP1A2CYP3A4
SCHEMBL11853062 0.82 NAMPT (0.44) NAMPTUSP2LMNACYP2C9CYP2C19
SCHEMBL26148108 0.80 TSHR (0.40) TSHRHSD17B10HDAC3HDAC1HDAC2
SCHEMBL13188656 0.80 CYP4A11 (0.51) LMNACYP2C9CYP2C19CYP1A2CYP3A4
SCHEMBL20862455 0.76 MAOA (0.40) HDAC3HDAC1HDAC2NCOR2
SCHEMBL10084755 0.76 MTNR1A (0.52) CYP2C9CYP2C19CYP1A2CYP3A4MEN1
SCHEMBL4453600 0.76 LTB4R (0.55) LMNAMAPT

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5338738-A Cerebral function enhancers: acyclic amide derivatives of pyrimidinylpiperidines BRISTOL-MYERS SQUIBB COMPANY (US) 1994-08-16 US disclosed