SCHEMBL9348479

SCHEMBL9348479

COc1c(OC)c(OC)c2c(=O)c3cccc(OCc4ccccc4)c3[nH]c2c1OC

nearest known ligand 0.48

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ADORA3 P0DMS8 1/20 0.48
CTSV O60911 2/20 0.46
CTSL P07711 2/20 0.46
PIK3CG P48736 1/20 0.44
MAPT P10636 2/20 0.43
KDM4E B2RXH2 1/20 0.43
MEN1 O00255 1/20 0.43
LMNA P02545 1/20 0.43
POLB P06746 1/20 0.43
BLM P54132 1/20 0.43
KMT2A Q03164 1/20 0.43
MCL1 Q07820 1/20 0.43
MAPK1 P28482 1/20 0.41
TDP1 Q9NUW8 1/20 0.41
L3MBTL1 Q9Y468 1/20 0.41
ABCG2 Q9UNQ0 2/20 0.41
LTA4H P09960 1/20 0.41
PLA2G2A P14555 1/20 0.41
TRPM8 Q7Z2W7 1/20 0.41
ALDH1A1 P00352 2/20 0.40

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9348380 0.88 CTSV (0.44) ADORA3CTSVCTSLMAPTKDM4E
SCHEMBL9348686 0.77 CTSV (0.41) ADORA3CTSVCTSLMAPTKDM4E
SCHEMBL9348689 0.76 CTSV (0.39) ADORA3CTSVCTSLMAPTKDM4E
SCHEMBL9352534 0.75 CTSV (0.51) ADORA3CTSVCTSLMAPTKDM4E
SCHEMBL5879271 0.74 ADORA3 (0.53) ADORA3CTSVCTSLPIK3CGMAPT
SCHEMBL8769400 0.73 PRKCA (0.52) ADORA3PIK3CGMAPTMEN1KMT2A
SCHEMBL17912878 0.71 MAPT (0.66) MAPTMAPK1TDP1L3MBTL1ABCG2
SCHEMBL16107056 0.70 ALDH1A1 (0.50) ADORA3CTSVCTSLPIK3CGMAPT
SCHEMBL11115687 0.70 MAPT (0.60) ADORA3CTSVCTSLPIK3CGMAPT
SCHEMBL14376020 0.70 KDM4E (0.44) CTSVMAPTKDM4EMEN1LMNA

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-1992016509-A1 MULTISUBSTITUTED 1-HYDROXY-9-ACRIDONES WITH ANTICANCER ACTIVITY SLOAN-KETTERING INSTITUTE FOR CANCER RESEARCH (US) 1992-10-01 WO claimed
US-5296602-A Condensing substituted ortho-halo- or ortho-aminobenzoic acid with meta-halo- or meta-aminoanisole, cyclizing, N-alkylating, de-O-methylating SLOAN-KETTERING INSTITUTE FOR CANCER RESEARCH (US) 1994-03-22 US disclosed
WO-1992016509-A1 MULTISUBSTITUTED 1-HYDROXY-9-ACRIDONES WITH ANTICANCER ACTIVITY SLOAN-KETTERING INSTITUTE FOR CANCER RESEARCH (US) 1992-10-01 WO disclosed