SCHEMBL8769400

SCHEMBL8769400

O=C1NC(=O)c2c1c1c3cccc(OCc4ccccc4)c3[nH]c1c1[nH]c3c(OCc4ccccc4)cccc3c21

nearest known ligand 0.52

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
PRKCA P17252 2/20 0.52
EGFR P00533 1/20 0.52
CHEK1 O14757 3/20 0.50
CDK4 P11802 9/20 0.49
CCND1 P24385 9/20 0.49
ADORA3 P0DMS8 1/20 0.49
CCNE2 O96020 5/20 0.49
CCNE1 P24864 5/20 0.49
CDK2 P24941 5/20 0.49
CAMK2B Q13554 4/20 0.49
CAMK2G Q13555 4/20 0.49
CAMK2D Q13557 4/20 0.49
CAMK2A Q9UQM7 4/20 0.49
PRKACA P17612 3/20 0.49
PRKACG P22612 3/20 0.49
PRKACB P22694 3/20 0.49
CCNB2 O95067 2/20 0.49
CDK1 P06493 2/20 0.49
CCNB1 P14635 2/20 0.49
CCNB3 Q8WWL7 2/20 0.49

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8314297 0.81 NQO1 (0.47) PRKCACHEK1ADORA3MAPTPIK3CG
SCHEMBL5879271 0.80 ADORA3 (0.53) CHEK1ADORA3MAPTPIK3CGLTA4H
SCHEMBL8599835 0.75 MAOA (0.54) CDK4CCND1CCNB2CDK1CCNB1
SCHEMBL27777168 0.73 SRD5A2 (0.56) ADORA3MAPTPIK3CGLTA4HPLA2G2A
SCHEMBL7284065 0.73 PIK3CG (0.47) EGFRADORA3MAPTPIK3CGLTA4H
SCHEMBL9348479 0.73 ADORA3 (0.48) ADORA3MEN1MAPTKMT2APIK3CG
SCHEMBL11115687 0.71 MAPT (0.60) ADORA3MEN1MAPTKMT2APIK3CG
SCHEMBL23887763 0.70 LTA4H (0.54) ADORA3MAPTKMT2APIK3CGLTA4H
SCHEMBL8123086 0.69 PRKCA (0.66) PRKCAEGFRCHEK1CDK4CCND1
SCHEMBL22566996 0.69 CDK4 (0.83) PRKCAEGFRCHEK1CDK4CCND1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0528030-B1 ANTITUMOR BE-13793C DERIVATIVE BANYU PHARMA CO LTD (JP) 1997-09-17 EP disclosed
US-5536827-A ANTITUMOR BANYU PHARMACEUTICAL CO., LTD. (JP) 1996-07-16 US disclosed
US-5478813-A Antitumor substance BE-13793C derivatives BANYU PHARMACEUTICAL CO., LTD. (JP) 1995-12-26 US disclosed
EP-0528030-A1 ANTITUMOR BE-13793C DERIVATIVE BANYU PHARMACEUTICAL CO., LTD. (JP) 1993-02-24 EP disclosed