SCHEMBL9360265

SCHEMBL9360265

Fc1cc(Br)cc(Sc2ccc3ccccc3c2)c1

nearest known ligand 0.48

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CYP2A6 P11509 3/20 0.48
CYP1A2 P05177 2/20 0.48
LMNA P02545 2/20 0.41
SMN1; SMN2 Q16637 1/20 0.41
MAP2K2 P36507 2/20 0.38
MAP2K1 Q02750 2/20 0.38
HAO1 Q9UJM8 1/20 0.38
SIRT2 Q8IXJ6 1/20 0.37
SIRT1 Q96EB6 1/20 0.37
SIRT3 Q9NTG7 1/20 0.37
ANPEP P15144 1/20 0.35
G6PD P11413 1/20 0.34
CCR6 P51684 1/20 0.34
HKDC1 Q2TB90 1/20 0.34
KDM4E B2RXH2 1/20 0.34
MAPT P10636 1/20 0.34
PKM P14618 1/20 0.34
MAPK1 P28482 1/20 0.34
KMT2A Q03164 1/20 0.34
MCL1 Q07820 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9458604 0.79 CYP2A6 (0.40) CYP2A6CYP1A2LMNASMN1; SMN2MAP2K2
SCHEMBL9361125 0.78 CYP2A6 (0.56) CYP2A6LMNASMN1; SMN2MAP2K2MAP2K1
SCHEMBL30832956 0.77 LMNA (0.57) CYP2A6CYP1A2LMNASMN1; SMN2MAP2K2
SCHEMBL761802 0.77 LMNA (0.57) CYP2A6CYP1A2LMNASMN1; SMN2MAP2K2
SCHEMBL9458698 0.73 CYP2A6 (0.46) CYP2A6CYP1A2LMNASMN1; SMN2MAP2K2
SCHEMBL18518053 0.71 CYP1A2 (0.52) CYP2A6CYP1A2SMN1; SMN2KDM4EMAPT
SCHEMBL15207756 0.71 MAOA (0.47) CYP2A6LMNASMN1; SMN2HAO1MAPT
SCHEMBL9458067 0.71 PTGIR (0.35) LMNASMN1; SMN2MAPTMAPK1KMT2A
SCHEMBL3281214 0.71 LMNA (0.52) CYP2A6CYP1A2LMNASMN1; SMN2MAP2K2
SCHEMBL11300299 0.70 ALDH1A1 (0.50) CYP2A6CYP1A2LMNASMN1; SMN2MAP2K2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 8 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0409412-B1 Diaryl ether cyclic ethers ICI PLC (GB) 1994-07-20 EP disclosed
EP-0409414-B1 DIARYL ETHER CYCLOALKANES IMPERIAL CHEMICAL INDUSTRIES PLC (GB) 1993-09-29 EP disclosed
US-5214070-A Lipoxygenase inhibitors IMPERIAL CHEMICAL INDUSTRIES PLC (GB) 1993-05-25 US disclosed
US-5208259-A Lipoxygenase enzyme inhibitors IMPERIAL CHEMICAL INDUSTRIES (GB) 1993-05-04 US disclosed
US-5137913-A Inhibitors of the enzyme 5-lipoxygenase IMPERIAL CHEMICAL INDUSTRIES PLC (GB) 1992-08-11 US disclosed
EP-0409413-A2 Diaryl ether heterocycles IMPERIAL CHEMICAL INDUSTRIES PLC (GB) 1991-01-23 EP disclosed
EP-0409414-A1 Diaryl ether cycloalkanes IMPERIAL CHEMICAL INDUSTRIES PLC (GB) 1991-01-23 EP disclosed
EP-0409412-A2 Diaryl ether cyclic ethers IMPERIAL CHEMICAL INDUSTRIES PLC (GB) 1991-01-23 EP disclosed