SCHEMBL9364266

SCHEMBL9364266

CCCCOC(=O)OC1=C(C)N(C)C(C)=C(OC(=O)OCCCC)C1c1ccc(Br)cc1

nearest known ligand 0.41

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
SMN1; SMN2 Q16637 2/20 0.41
HPGD P15428 2/20 0.41
NPSR1 Q6W5P4 2/20 0.41
GAA P10253 2/20 0.40
KDM4E B2RXH2 2/20 0.40
HTT P42858 3/20 0.39
TSHR P16473 3/20 0.38
TP53 P04637 1/20 0.38
ELANE P08246 1/20 0.37
MGLL Q99685 1/20 0.36
ATM Q13315 1/20 0.36
HRH2 P25021 1/20 0.35
HRH1 P35367 1/20 0.35
HRH3 Q9Y5N1 3/20 0.35
HSD17B10 Q99714 1/20 0.35
LMNA P02545 3/20 0.35
MAPT P10636 2/20 0.35
ALDH1A1 P00352 1/20 0.35
CACNA1F O60840 1/20 0.35
BCHE P06276 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9364315 0.93 NPSR1 (0.42) SMN1; SMN2HPGDNPSR1GAAKDM4E
SCHEMBL9368993 0.84 ADORA3 (0.45) SMN1; SMN2MGLLHRH2HRH1LMNA
SCHEMBL9118263 0.81 NPSR1 (0.59) SMN1; SMN2HPGDNPSR1GAAKDM4E
SCHEMBL9367544 0.81 TSHR (0.47) SMN1; SMN2HPGDNPSR1KDM4EHTT
SCHEMBL9369053 0.79 ALDH1A1 (0.39) SMN1; SMN2HPGDLMNAMAPTALDH1A1
SCHEMBL9364303 0.78 HPGD (0.40) SMN1; SMN2HPGDNPSR1GAAKDM4E
SCHEMBL9363815 0.76 NPSR1 (0.48) SMN1; SMN2HPGDNPSR1GAAKDM4E
SCHEMBL9364038 0.76 PKM (0.47) NPSR1GAAKDM4EHTTTSHR
SCHEMBL9364015 0.74 HSP90AA1 (0.42) SMN1; SMN2HPGDNPSR1GAAKDM4E
SCHEMBL9364030 0.74 HPGD (0.43) SMN1; SMN2HPGDNPSR1GAAKDM4E

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0451654-B1 Use of N-alkylated 1,4-dihydropyridine carboxylic acid esters as drugs, new compounds and process for their preparation BAYER AG (DE) 1994-09-07 EP claimed
EP-0451654-A2 Use of N-alkylated 1,4-dihydropyridine carboxylic acid esters as drugs, new compounds and process for their preparation BAYER AG (DE) 1991-10-16 EP claimed
EP-0451654-B1 Use of N-alkylated 1,4-dihydropyridine carboxylic acid esters as drugs, new compounds and process for their preparation BAYER AG (DE) 1994-09-07 EP disclosed
EP-0451654-A2 Use of N-alkylated 1,4-dihydropyridine carboxylic acid esters as drugs, new compounds and process for their preparation BAYER AG (DE) 1991-10-16 EP disclosed