SCHEMBL9364669

SCHEMBL9364669

CC(C)(C)OC(=O)NC(C(=O)O)c1ccc2ncsc2c1

nearest known ligand 0.43

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
IRAK4 Q9NWZ3 2/20 0.43
NPC1 O15118 3/20 0.43
RAB9A P51151 3/20 0.43
KDM4E B2RXH2 2/20 0.43
HKDC1 Q2TB90 1/20 0.43
TDP1 Q9NUW8 1/20 0.43
L3MBTL1 Q9Y468 1/20 0.43
TAS1R3 Q7RTX0 1/20 0.41
TAS1R1 Q7RTX1 1/20 0.41
FFAR1 O14842 1/20 0.40
CTSS P25774 1/20 0.40
CTSK P43235 1/20 0.40
S1PR3 Q99500 2/20 0.39
MEN1 O00255 2/20 0.39
KMT2A Q03164 2/20 0.39
POLB P06746 1/20 0.39
NTRK1 P04629 2/20 0.38
NTRK2 Q16620 2/20 0.38
OGA O60502 2/20 0.38
LMNA P02545 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8977487 0.80 RAB9A (0.49) NPC1RAB9AL3MBTL1LMNA
SCHEMBL8977464 0.79 LCK (0.54) NPC1RAB9AMEN1KMT2ALMNA
SCHEMBL10926694 0.79 CTSS (0.41) KDM4ECTSSCTSKS1PR3
SCHEMBL10627562 0.78 CTSS (0.43) NPC1RAB9AKDM4ETDP1CTSS
SCHEMBL10631857 0.77 ALDH1A1 (0.45) NPC1RAB9ATAS1R3TAS1R1CTSS
SCHEMBL11121473 0.76 CTSS (0.41) CTSSCTSKS1PR3
SCHEMBL25382759 0.75 NPC1 (0.51) IRAK4NPC1RAB9AKDM4EHKDC1
SCHEMBL30554088 0.75 NPC1 (0.51) IRAK4NPC1RAB9AKDM4EHKDC1
SCHEMBL9619945 0.75 CTSS (0.38) NPC1RAB9ACTSSCTSKS1PR3
SCHEMBL10725965 0.75 YARS1 (0.47) KDM4ETDP1CTSSCTSKMEN1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0292806-B1 Substituted vinyl cephalosporins, process for their preparation and their use as medicines BAYER AG (DE) 1994-11-02 EP disclosed
US-5171854-A Antibiotics BAYER AKTIENGESELLSCHAFT (DE) 1992-12-15 US disclosed
EP-0292806-A2 Substituted vinyl cephalosporins, process for their preparation and their use as medicines BAYER AG (DE) 1988-11-30 EP disclosed