SCHEMBL9619945

SCHEMBL9619945

CC(C)(C)OC(=O)NC(C(=O)O)c1ccc2sc(N)nc2c1

nearest known ligand 0.42

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CTSS P25774 1/20 0.38
CTSK P43235 1/20 0.38
NPC1 O15118 2/20 0.38
RAB9A P51151 2/20 0.38
SCN4A P35499 1/20 0.38
SMN1; SMN2 Q16637 1/20 0.38
LIPG Q9Y5X9 1/20 0.37
DYRK1A Q13627 1/20 0.36
S1PR3 Q99500 2/20 0.36
FTO Q9C0B1 1/20 0.36
KIT P10721 1/20 0.35
HDAC3 O15379 2/20 0.35
HDAC1 Q13547 2/20 0.35
HDAC2 Q92769 2/20 0.35
HDAC8 Q9BY41 2/20 0.35
HDAC6 Q9UBN7 2/20 0.35
HDAC4 P56524 1/20 0.35
HDAC7 Q8WUI4 1/20 0.35
HDAC10 Q969S8 1/20 0.35
HDAC11 Q96DB2 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8977487 0.91 RAB9A (0.49) NPC1RAB9ASCN4ASMN1; SMN2LIPG
SCHEMBL10627562 0.79 CTSS (0.43) CTSSCTSKNPC1RAB9AS1PR3
SCHEMBL10627574 0.77 CTSS (0.40) CTSSCTSKNPC1RAB9AS1PR3
Bromide SCHEMBL9620176 0.77 CTSS (0.40) CTSSCTSKS1PR3PIK3CAPIK3CD
SCHEMBL8977464 0.77 LCK (0.54) NPC1RAB9ASMN1; SMN2HDAC3HDAC1
SCHEMBL11121473 0.77 CTSS (0.41) CTSSCTSKS1PR3GABRB1GABRB2
SCHEMBL3375087 0.75 CTSK (0.51) CTSSCTSKS1PR3GABRB1GABRB2
SCHEMBL3375084 0.75 CTSK (0.51) CTSSCTSKS1PR3GABRB1GABRB2
SCHEMBL9364669 0.75 IRAK4 (0.43) CTSSCTSKNPC1RAB9AS1PR3
SCHEMBL9620010 0.75 CTSS (0.43) CTSSCTSKS1PR3ALDH1A1PPARA

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-RE33948-E Bactericides, animal growth regulators BAYER AKTIENGESELLSCHAFT (DE) 1992-06-02 US disclosed
US-4748163-A Novel β-lactam antibiotics BAYER AKTIENGESELLSCHAFT (DE) 1988-05-31 US disclosed
EP-0195947-A2 Beta-lactam antibiotics, process for their preparation and their use as and in medicaments BAYER AG (DE) 1986-10-01 EP disclosed