SCHEMBL9368243

SCHEMBL9368243

O=C(c1cccnc1)c1ccc2[nH]c(=O)oc2c1

nearest known ligand 0.53

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 4/20 0.53
CREBBP Q92793 1/20 0.53
KDM4E B2RXH2 1/20 0.53
PDE3B Q13370 2/20 0.49
PDE3A Q14432 2/20 0.49
MAP2K1 Q02750 1/20 0.48
SMYD3 Q9H7B4 1/20 0.47
NOS1 P29475 1/20 0.44
ESR1 P03372 1/20 0.43
JAK3 P52333 1/20 0.42
APP P05067 1/20 0.41
GAA P10253 1/20 0.41
HCAR3 P49019 1/20 0.41
HCAR2 Q8TDS4 1/20 0.41
OGT O15294 1/20 0.41
SYK P43405 1/20 0.41
F7 P08709 1/20 0.41
F3 P13726 1/20 0.41
SARM1 Q6SZW1 1/20 0.41
SIRT2 Q8IXJ6 1/20 0.41

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6647933 0.84 ALDH1A1 (0.60) ALDH1A1CREBBPKDM4EPDE3BPDE3A
SCHEMBL17260664 0.77 KDM4E (0.62) ALDH1A1CREBBPKDM4ESMYD3NOS1
SCHEMBL14565010 0.76 NOS1 (0.52) ALDH1A1CREBBPKDM4ESMYD3NOS1
SCHEMBL9682938 0.76 TOP2A (0.51) ALDH1A1CREBBPKDM4EPDE3BPDE3A
SCHEMBL858860 0.76 CREBBP (0.48) ALDH1A1CREBBPKDM4EPDE3BPDE3A
SCHEMBL9484144 0.76 MAP2K1 (0.48) ALDH1A1PDE3BPDE3AMAP2K1ESR1
SCHEMBL9470246 0.75 MAP2K1 (0.47) ALDH1A1MAP2K1JAK3APPGAA
SCHEMBL29771053 0.75 KDM4E (0.67) ALDH1A1CREBBPKDM4EPDE3BPDE3A
SCHEMBL118684 0.75 KDM4E (0.67) ALDH1A1CREBBPKDM4EPDE3BPDE3A
SCHEMBL30494348 0.74 PDE3B (0.70) ALDH1A1PDE3BPDE3ANOS1OGT

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0463944-B1 Acylbenzoxazolinones, process for their preparation and pharmaceutical compositions containing them ADIR (FR) 1994-10-05 EP disclosed
US-5147883-A Antiischemic, stroke ADIR ET COMPAGNIE (FR) 1992-09-15 US disclosed
EP-0463944-A1 Acylbenzoxazolinones, process for their preparation and pharmaceutical compositions containing them ADIR ET COMPAGNIE (FR) 1992-01-02 EP disclosed