SCHEMBL9375402

SCHEMBL9375402

Brc1cccc(-c2nncc3ncccc23)c1

nearest known ligand 0.51

Predicted protein targets (top 19)

geneUniProtsupporting neighboursconfidence
GABRG2 P18507 9/20 0.43
GABRB3 P28472 9/20 0.43
GABRA5 P31644 9/20 0.43
GABRA3 P34903 9/20 0.43
GABRA1 P14867 7/20 0.43
IDO1 P14902 2/20 0.43
TDO2 P48775 1/20 0.43
BIRC5 O15392 1/20 0.40
CYP1A2 P05177 1/20 0.39
CYP2C19 P33261 1/20 0.39
HTT P42858 1/20 0.39
BCHE P06276 1/20 0.38
ACHE P22303 1/20 0.38
ALDH1A1 P00352 2/20 0.37
MEN1 O00255 1/20 0.37
KMT2A Q03164 1/20 0.37
NPSR1 Q6W5P4 1/20 0.37
LMNA P02545 1/20 0.37
EGFR P00533 1/20 0.37

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9376993 0.79 DYRK1A (0.51) CYP1A2
SCHEMBL9378645 0.78 GABRG2 (0.44) GABRG2GABRB3GABRA5GABRA3GABRA1
SCHEMBL9376329 0.74 MAPT (0.44) HTTALDH1A1MEN1KMT2ANPSR1
SCHEMBL28020925 0.71 IDO1 (0.48) IDO1TDO2BIRC5CYP1A2CYP2C19
SCHEMBL7362648 0.70 CAMKK2 (0.47) ALDH1A1MEN1KMT2AEGFR
SCHEMBL21805047 0.69 IDO1 (0.47) IDO1TDO2BIRC5BCHEACHE
SCHEMBL30088096 0.69 IDO1 (0.47) IDO1TDO2BIRC5BCHEACHE
SCHEMBL15606489 0.68 CYP2A6 (0.56) IDO1TDO2BIRC5BCHEACHE
SCHEMBL31070756 0.68 CYP2A6 (0.56) IDO1TDO2BIRC5BCHEACHE
SCHEMBL19051830 0.67 ALDH1A1 (0.44) IDO1TDO2BIRC5CYP1A2ALDH1A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0612321-A1 PYRIDO PYRIDAZINONE AND PYRIDAZINTHIONE COMPOUNDS WITH PDE IV INHIBITING ACTIVITY SYNTEX (U.S.A.) INC. (US) 1994-08-31 EP disclosed