SCHEMBL9375907

SCHEMBL9375907

CC1(C)C(=O)Nc2ccc(C(=O)Nc3ccc(C#N)cc3)cc21

nearest known ligand 0.50

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
PGR P06401 4/20 0.50
CYP26A1 O43174 2/20 0.48
CYP3A4 P08684 2/20 0.48
RARA P10276 2/20 0.48
MLYCD O95822 1/20 0.47
MEN1 O00255 2/20 0.46
KMT2A Q03164 2/20 0.46
NPC1 O15118 1/20 0.46
RAB9A P51151 1/20 0.46
RPS6KA2 Q15349 1/20 0.46
TLK2 Q86UE8 1/20 0.46
ESR1 P03372 1/20 0.46
NAMPT P43490 2/20 0.45
MAPKAPK2 P49137 1/20 0.45
LMNA P02545 2/20 0.43
POLB P06746 1/20 0.43
SMN1; SMN2 Q16637 1/20 0.43
SIRT2 Q8IXJ6 1/20 0.43
ROCK2 O75116 1/20 0.43
ALDH1A1 P00352 1/20 0.43

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9840448 0.91 CYP26A1 (0.48) CYP26A1CYP3A4RARAMLYCDMEN1
SCHEMBL9380846 0.84 BACE1 (0.52) CYP26A1CYP3A4RARAMEN1KMT2A
SCHEMBL9382115 0.84 CYP26A1 (0.53) PGRCYP26A1CYP3A4RARAMEN1
SCHEMBL9380134 0.82 RAB9A (0.57) CYP3A4MEN1KMT2ANPC1RAB9A
SCHEMBL9865366 0.78 MAPT (0.52) PGRCYP3A4MEN1KMT2ARAB9A
SCHEMBL25944404 0.77 PGR (0.71) PGR
SCHEMBL9375803 0.76 MAPT (0.45) CYP26A1CYP3A4RARAMEN1KMT2A
SCHEMBL9380149 0.76 PRKAA2 (0.44) MEN1KMT2ANPC1RAB9ATLK2
SCHEMBL9376618 0.76 RARB (0.56) CYP26A1CYP3A4RARAMLYCDMEN1
SCHEMBL9375391 0.75 CYP26A1 (0.52) PGRCYP26A1CYP3A4RARAMEN1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0344634-B1 Bicyclic carboxamides, process for their preparation and medicaments containing them BOEHRINGER MANNHEIM GMBH (DE) 1994-03-30 EP disclosed
US-5019587-A Anticoagulants BOEHRINGER MANNHEIM GMBH (DE) 1991-05-28 US disclosed
EP-0344634-A1 Bicyclic carboxamides, process for their preparation and medicaments containing them Roche Diagnostics GmbH (DE) 1989-12-06 EP disclosed