Cyclopentane

Cyclopentane

SCHEMBL9375968

C1CCCC1.NC(=O)NO

nearest known ligand 0.77

Full drug profile on Sugi Atlas →

Known targets — ChEMBL curated mechanism

RRM1RRM2RRM2B

The experimentally established mechanism targets of Cyclopentane. The predicted profile below is derived independently by chemical similarity — agreement is a validation signal, a miss is honest.

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
LMNA P02545 4/20 0.77
TSHR P16473 2/20 0.77
NFKB1 P19838 2/20 0.77
CA2 P00918 2/20 0.77
BLM P54132 2/20 0.77
PMP22 Q01453 2/20 0.77
CYP3A4 P08684 2/20 0.77
CA5A P35218 1/20 0.77
CA9 Q16790 1/20 0.77
CYP1A2 P05177 1/20 0.44
MAOA P21397 1/20 0.44
MAOB P27338 1/20 0.44
THPO P40225 1/20 0.44
HDAC8 Q9BY41 1/20 0.41
HDAC6 Q9UBN7 1/20 0.41
ALDH1A1 P00352 3/20 0.36
TDP1 Q9NUW8 2/20 0.36
OR51E2 Q9H255 1/20 0.36
KDM4E B2RXH2 2/20 0.35
PTGS1 P23219 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
Hydroxyurea SCHEMBL9377620 1.00
Hydroxyurea SCHEMBL10966425 1.00
Hydroxyurea SCHEMBL5329855 0.88 LMNA (1.00) LMNATSHRNFKB1CA2BLM
Hydroxyurea SCHEMBL4004 0.88
Hydroxyurea SCHEMBL93814 0.88 LMNA (1.00) LMNATSHRNFKB1CA2BLM
Hydroxyurea SCHEMBL23274911 0.84
Hydroxyurea SCHEMBL306433 0.84
Hydroxyurea SCHEMBL28868410 0.84
Hydroxyurea SCHEMBL15011410 0.84
Hydroxyurea SCHEMBL308240 0.84

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0150040-B1 Imidazodiazepine derivatives HOFFMANN LA ROCHE (CH) 1994-08-31 EP disclosed
EP-0150040-A2 Imidazodiazepine derivatives F. HOFFMANN-LA ROCHE AG (CH) 1985-07-31 EP disclosed