SCHEMBL9397293

SCHEMBL9397293

N=C=O.Oc1ccnc2cc(Br)ccc12

nearest known ligand 0.45

Predicted protein targets (top 19)

geneUniProtsupporting neighboursconfidence
SLC22A12 Q96S37 6/20 0.45
ALK Q9UM73 1/20 0.43
CYP1A2 P05177 1/20 0.39
CYP2C19 P33261 1/20 0.39
HTT P42858 1/20 0.39
GAK O14976 1/20 0.37
PTGES O14684 1/20 0.36
KDM4E B2RXH2 1/20 0.35
ALDH1A1 P00352 1/20 0.35
SMN1; SMN2 Q16637 1/20 0.35
PREP P48147 1/20 0.35
PLAU P00749 2/20 0.35
PLG P00747 1/20 0.35
PLAT P00750 1/20 0.35
ERN1 O75460 1/20 0.34
EGFR P00533 1/20 0.34
CES2 O00748 1/20 0.33
GALR3 O60755 1/20 0.33
ALOX15 P16050 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL1490718 0.90 ALK (0.50) SLC22A12ALKCYP1A2CYP2C19HTT
SCHEMBL9397259 0.81 GAK (0.37) CYP1A2GAKERN1
SCHEMBL360254 0.75 SLC22A12 (0.51) SLC22A12ALKCYP1A2CYP2C19HTT
SCHEMBL23498024 0.73 SLC22A12 (0.37) SLC22A12ALKCYP2C19GAKKDM4E
SCHEMBL4470963 0.71 ALK (0.53) SLC22A12ALKCYP1A2CYP2C19HTT
SCHEMBL28164080 0.71 TLR8 (0.54) HTTKDM4EALDH1A1SMN1; SMN2EGFR
SCHEMBL29509132 0.71 TLR8 (0.54) HTTKDM4EALDH1A1SMN1; SMN2EGFR
SCHEMBL29896720 0.71 ALK (0.53) SLC22A12ALKCYP1A2CYP2C19HTT
SCHEMBL30135541 0.70 SLC22A12 (0.50) SLC22A12ALKKDM4EALDH1A1SMN1; SMN2
SCHEMBL7374970 0.70 SLC22A12 (0.50) SLC22A12ALKKDM4EALDH1A1SMN1; SMN2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5344922-A 4-hydroxyquinaldic acid derivatives BOARD OF REGENTS, UNIVERSITY OF TEXAS 1994-09-06 US disclosed
US-5028707-A 4-hydroxyquinaldic acid derivatives BOARD OF REGENTS, UNIVERSITY OF TEXAS (US) 1991-07-02 US disclosed
WO-1991007390-A1 4-HYDROXYQUINALDIC ACID DERIVATIVES BOARD OF REGENTS, THE UNIVERSITY OF TEXAS SYSTEM (US) 1991-05-30 WO disclosed