SCHEMBL9400933

SCHEMBL9400933

O=C1c2ccccc2C(=O)N1CC(O)CN1CCN(c2ncccn2)CC1

nearest known ligand 0.66

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
HTR1A P08908 7/20 0.63
ALDH1A1 P00352 4/20 0.49
POLB P06746 2/20 0.49
LMNA P02545 1/20 0.49
MAPT P10636 1/20 0.49
HPGD P15428 1/20 0.49
MAPK1 P28482 1/20 0.49
SMN1; SMN2 Q16637 1/20 0.49
HSD17B10 Q99714 1/20 0.49
KDM4E B2RXH2 1/20 0.48
DRD2 P14416 2/20 0.47
HTR2A P28223 2/20 0.47
HTR7 P34969 2/20 0.47
HTR6 P50406 2/20 0.47
DRD3 P35462 3/20 0.47
MEN1 O00255 1/20 0.46
KMT2A Q03164 1/20 0.46
ABCB11 O95342 1/20 0.46
CYP1A2 P05177 1/20 0.46
ADRA2A P08913 1/20 0.46

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL11104845 0.89 ALDH1A1 (0.63) ALDH1A1POLBLMNAMAPTHPGD
SCHEMBL9401026 0.87 HTR1A (0.52) HTR1AALDH1A1POLBLMNAMAPT
SCHEMBL9400979 0.83 HTR1A (0.47) HTR1AALDH1A1LMNAMAPTSMN1; SMN2
SCHEMBL9400890 0.81 KMT2A (0.55) HTR1AALDH1A1MAPK1KDM4EDRD2
SCHEMBL11114070 0.80 HTR1A (0.67) HTR1AALDH1A1POLBLMNAMAPT
SCHEMBL9481460 0.80 HTR1A (0.68) HTR1AALDH1A1LMNAMAPTHPGD
SCHEMBL17861450 0.80 SORD (0.50) HTR1AALDH1A1POLBLMNAMAPT
SCHEMBL11106525 0.80 HTR1A (0.53) HTR1AKDM4EDRD2MEN1KMT2A
SCHEMBL11114528 0.80 HTR1A (0.50) HTR1AALDH1A1POLBLMNAMAPT
SCHEMBL9401013 0.80 HTR1A (0.84) HTR1AALDH1A1DRD2HTR2AHTR7

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 8 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5314884-A Antidepressants, anxiolytic agents TROPONWERKE GMBH & CO. (DE) 1994-05-24 US disclosed
US-5187276-A Anxiolytics, neuroleptics, antidepressants, and nootropic agents TROPONWERKE GMBH & CO. KG. (DE) 1993-02-16 US disclosed
US-4988809-A CENTRAL NERVOUS SYSTEM TROPONWERKE GMBH & CO., KG (DE) 1991-01-29 US disclosed
EP-0129128-B1 2-PYRIMIDINYL-1-PIPERAZINE DERIVATIVES, PROCESS FOR THEIR PREPARATION AND MEDICINES CONTAINING THEM Troponwerke GmbH & Co. KG (DE) 1990-11-22 EP disclosed
US-4937343-A NEUROLEPTICS OR ANTIDEPRESSANTS TROPONWERKE GMBH & CO. KG (DE) 1990-06-26 US disclosed
US-4818756-A CENTRAL NERVOUS SYSTEM DISORDERS TROPONWERKE GMBH & CO., KG (DE) 1989-04-04 US disclosed
EP-0129128-A2 2-Pyrimidinyl-1-piperazine derivatives, process for their preparation and medicines containing them Troponwerke GmbH & Co. KG (DE) 1984-12-27 EP disclosed
US-4479954-A ANTIDIABETIC AGENTS EISAI CO., LTD. (JP) 1984-10-30 US disclosed