SCHEMBL9401014

SCHEMBL9401014

Fc1cccc(Cl)c1-c1cnc(N2CCNCC2)nc1

nearest known ligand 0.47

Predicted protein targets (top 16)

geneUniProtsupporting neighboursconfidence
INPPL1 O15357 2/20 0.47
HTR1A P08908 1/20 0.46
SLC6A2 P23975 1/20 0.46
TAAR1 Q96RJ0 1/20 0.45
FEN1 P39748 1/20 0.44
CNR2 P34972 1/20 0.44
KDM4E B2RXH2 2/20 0.44
ALDH1A1 P00352 1/20 0.44
ADRB1 P08588 2/20 0.43
DRD2 P14416 1/20 0.43
DRD3 P35462 1/20 0.43
L3MBTL1 Q9Y468 1/20 0.42
BCL6 P41182 1/20 0.41
CHRNB2 P17787 1/20 0.41
CHRNA4 P43681 1/20 0.41
SCN9A Q15858 1/20 0.40

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9400916 0.78 SIGMAR1 (0.44) HTR1AKDM4EDRD2DRD3
SCHEMBL9400962 0.77 SIGMAR1 (0.46) HTR1AKDM4EDRD2DRD3L3MBTL1
Hydrochloric Acid SCHEMBL10568101 0.76 SIGMAR1 (0.45) HTR1AKDM4EDRD2DRD3
SCHEMBL9400931 0.74 ALDH1A1 (0.55) KDM4EALDH1A1L3MBTL1
SCHEMBL5787773 0.74 ALDH1A1 (0.63) KDM4EALDH1A1ADRB1L3MBTL1
Hydrochloric Acid SCHEMBL5787470 0.73 ALDH1A1 (0.62) KDM4EALDH1A1ADRB1L3MBTL1
SCHEMBL9400849 0.72 HTR3A (0.54) INPPL1HTR1ATAAR1KDM4EALDH1A1
SCHEMBL6787637 0.72 HTR7 (0.54) HTR1ATAAR1FEN1KDM4EALDH1A1
SCHEMBL6782999 0.71 ADRB1 (0.53) INPPL1TAAR1FEN1CNR2KDM4E
SCHEMBL9400977 0.71 TAAR1 (0.64) HTR1ATAAR1KDM4EALDH1A1ADRB1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 7 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5314884-A Antidepressants, anxiolytic agents TROPONWERKE GMBH & CO. (DE) 1994-05-24 US disclosed
US-5187276-A Anxiolytics, neuroleptics, antidepressants, and nootropic agents TROPONWERKE GMBH & CO. KG. (DE) 1993-02-16 US disclosed
US-4988809-A CENTRAL NERVOUS SYSTEM TROPONWERKE GMBH & CO., KG (DE) 1991-01-29 US disclosed
EP-0129128-B1 2-PYRIMIDINYL-1-PIPERAZINE DERIVATIVES, PROCESS FOR THEIR PREPARATION AND MEDICINES CONTAINING THEM Troponwerke GmbH & Co. KG (DE) 1990-11-22 EP disclosed
US-4937343-A NEUROLEPTICS OR ANTIDEPRESSANTS TROPONWERKE GMBH & CO. KG (DE) 1990-06-26 US disclosed
US-4818756-A CENTRAL NERVOUS SYSTEM DISORDERS TROPONWERKE GMBH & CO., KG (DE) 1989-04-04 US disclosed
EP-0129128-A2 2-Pyrimidinyl-1-piperazine derivatives, process for their preparation and medicines containing them Troponwerke GmbH & Co. KG (DE) 1984-12-27 EP disclosed