SCHEMBL9402833

SCHEMBL9402833

CC(C)(C)C(=O)Nc1ccc(O)c(Cl)c1

nearest known ligand 0.60

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
L3MBTL1 Q9Y468 1/20 0.60
MAPT P10636 3/20 0.54
ALDH1A1 P00352 2/20 0.54
LMNA P02545 1/20 0.54
NR1H4 Q96RI1 3/20 0.50
NPSR1 Q6W5P4 1/20 0.50
CA12 O43570 1/20 0.50
CA1 P00915 1/20 0.50
CA2 P00918 1/20 0.50
CA7 P43166 1/20 0.50
CA9 Q16790 1/20 0.50
CA14 Q9ULX7 1/20 0.50
NPY2R P49146 4/20 0.49
HTT P42858 1/20 0.49
LCK P06239 1/20 0.49
CTSL P07711 1/20 0.49
PTPRC P08575 1/20 0.49
PTPN2 P17706 1/20 0.49
PTPN1 P18031 1/20 0.49
CTSS P25774 1/20 0.49

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL334142 0.86 L3MBTL1 (0.64) L3MBTL1MAPTLMNANPSR1CA2
SCHEMBL7757014 0.84 MAPT (0.51) MAPTALDH1A1LMNANR1H4CA2
SCHEMBL12662131 0.83 L3MBTL1 (0.60) L3MBTL1MAPTALDH1A1LMNACA2
SCHEMBL3788796 0.83 L3MBTL1 (0.60) L3MBTL1MAPTALDH1A1LMNANPSR1
SCHEMBL18701612 0.81 HTT (0.68) L3MBTL1MAPTALDH1A1LMNANPSR1
SCHEMBL31192562 0.81 MAPT (0.61) L3MBTL1MAPTALDH1A1LMNANPSR1
SCHEMBL22724808 0.81 MAPT (0.61) L3MBTL1MAPTALDH1A1LMNANPSR1
SCHEMBL9402610 0.80 GAA (0.59) L3MBTL1MAPTALDH1A1LMNANPSR1
SCHEMBL31198183 0.80 HSD17B10 (0.59) MAPTALDH1A1LMNANR1H4CA12
SCHEMBL5674663 0.80 HSD17B10 (0.59) MAPTALDH1A1LMNANR1H4CA12

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 15 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-3222620-B1 CYANOQUINOLINE DERIVATIVES TIANJIN HEMAY ONCOLOGY PHARMACEUTICAL CO LTD (CN) 2019-11-20 EP disclosed
US-10246443-B2 Cyanoquinoline derivatives TIANJIN HEMAY ONCOLOGY PHARMACEUTICAL CO., LTD. (CN) 2019-04-02 US disclosed
EP-3222620-A1 CYANOQUINOLINE DERIVATIVES TIANJIN HEMAY ONCOLOGY PHARMACEUTICAL CO., LTD. (CN) 2017-09-27 EP disclosed
US-20170226093-A1 CYANOQUINOLINE DERIVATIVES TIANJIN HEMAY ONCOLOGY PHARMACEUTICAL CO., LTD. (CN) 2017-08-10 US disclosed
US-9676724-B2 Cyanoquinoline derivatives TIANJIN HEMAY ONCOLOGY PHARMACEUTICAL CO., LTD. (CN) 2017-06-13 US disclosed
EP-2581372-B1 CYANOQUINOLINE DERIVATIVES TIANJIN HEMAY ONCOLOGY PHARMACEUTICAL CO LTD (CN) 2017-06-07 EP disclosed
US-20160185728-A1 CYANOQUINOLINE DERIVATIVES TIANJIN HEMAY ONCOLOGY PHARMACEUTICAL CO., LTD. (CN) 2016-06-30 US disclosed
US-9187458-B2 Cyanoquinoline derivatives TIANJIN HEMAY BIO-TECH CO., LTD. (CN) 2015-11-17 US disclosed
US-20130225579-A1 CYANOQUINOLINE DERIVATIVES TIANJIN HEMAY BIO-TECH CO., LTD. (CN) 2013-08-29 US disclosed
EP-2581372-A1 CYANOQUINOLINE DERIVATIVES Tianjin Hemay Bio-Tech Co., Ltd. (CN) 2013-04-17 EP disclosed
US-5371271-A Pesticides, fungicides BAYER AKTIENGESELLSCHAFT (DE) 1994-12-06 US disclosed
US-5260474-A Fungicides BAYER AKTIENGESELLSCHAFT (DE) 1993-11-09 US disclosed
EP-0293718-B1 SUBSTITUTED AMINOPHENYL CARBAMATE BAYER AG (DE) 1993-02-03 EP disclosed
US-4939170-A Substituted aminophenyl carbamates BAYER AKTIENGESELLSCHAFT (DE) 1990-07-03 US disclosed
EP-0293718-A2 Substituted aminophenyl carbamate BAYER AG (DE) 1988-12-07 EP disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (4 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-10246443-B2 Cyanoquinoline derivatives CBR3, CYP3A4, CDK1 L3MBTL1 1535/4885MAPT 43/4885ALDH1A1 2007/4885
US-20130225579-A1 CYANOQUINOLINE DERIVATIVES CBR3, CYP3A4, CDK1 L3MBTL1 1535/4885MAPT 43/4885ALDH1A1 2007/4885
US-20160185728-A1 CYANOQUINOLINE DERIVATIVES CBR3, CYP3A4, CDK1 L3MBTL1 1535/4885MAPT 43/4885ALDH1A1 2007/4885
US-20170226093-A1 CYANOQUINOLINE DERIVATIVES CBR3, CYP3A4, CDK1 L3MBTL1 1535/4885MAPT 43/4885ALDH1A1 2007/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.