SCHEMBL9404549

SCHEMBL9404549

CC(CCc1ccccc1)[C@@]1(n2cnc3c(N)nc(Cl)nc32)O[C@H](CO)[C@@H](O)[C@H]1O

nearest known ligand 0.44

Predicted protein targets (top 8)

geneUniProtsupporting neighboursconfidence
ADORA2A P29274 7/20 0.44
ADORA3 P0DMS8 7/20 0.43
ADORA1 P30542 6/20 0.43
PDE2A O00408 2/20 0.42
ADRA1A P35348 1/20 0.42
PDE4D Q08499 1/20 0.42
PDE3A Q14432 1/20 0.42
ADORA2B P29275 2/20 0.42

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7743876 0.78 ADORA2A (0.46) ADORA2AADORA3ADORA1ADORA2B
SCHEMBL859642 0.78 ADORA2A (0.46) ADORA2AADORA3ADORA1ADORA2B
SCHEMBL10709057 0.76 ADORA2A (0.48) ADORA2AADORA3ADORA1PDE2AADRA1A
SCHEMBL6538264 0.76 ADORA2A (0.57) ADORA2AADORA3ADORA1PDE2AADRA1A
SCHEMBL9494041 0.76 ADORA1 (0.46) ADORA1
SCHEMBL6829149 0.75 AHCY (0.43) ADORA2AADORA3ADORA1ADORA2B
SCHEMBL7793907 0.73 ADORA3 (0.61) ADORA2AADORA3ADORA1ADORA2B
SCHEMBL10710910 0.72 ADORA2A (0.46) ADORA2AADORA3ADORA1PDE2AADRA1A
SCHEMBL5525776 0.72 PI4KA (0.45) ADORA2AADORA3ADORA1ADORA2B
SCHEMBL13268818 0.72 PI4KA (0.45) ADORA2AADORA3ADORA1ADORA2B

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0603348-A1 PURINE DERIVATIVES NOVO NORDISK A/S (DK) 1994-06-29 EP claimed
WO-1993023418-A1 PURINE DERIVATIVES NOVO NORDISK A/S (DK) 1993-11-25 WO claimed