SCHEMBL9409382

SCHEMBL9409382

CCCN(Cc1ccc(-c2ccccc2C#N)cc1)Cc1[nH]ncc1C(=O)OCC

nearest known ligand 0.39

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
KDM4E B2RXH2 10/20 0.39
ALDH1A1 P00352 10/20 0.39
L3MBTL1 Q9Y468 9/20 0.39
TDP1 Q9NUW8 6/20 0.39
LMNA P02545 4/20 0.39
HPGD P15428 4/20 0.39
NPSR1 Q6W5P4 3/20 0.39
GPR55 Q9Y2T6 2/20 0.38
HTT P42858 1/20 0.38
CYP1A2 P05177 2/20 0.38
CYP3A4 P08684 2/20 0.38
CYP2C9 P11712 2/20 0.38
CYP2C19 P33261 2/20 0.38
MAPT P10636 3/20 0.38
HSD17B10 Q99714 2/20 0.37
ALOX15 P16050 1/20 0.37
SMN1; SMN2 Q16637 1/20 0.37
MEN1 O00255 4/20 0.37
KMT2A Q03164 4/20 0.37
TRPA1 O75762 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6611120 0.76 AGTR1 (0.55) ALDH1A1SMN1; SMN2
SCHEMBL8552171 0.76 MAP2K1 (0.40) KDM4EALDH1A1L3MBTL1TDP1LMNA
SCHEMBL10924590 0.75 ALDH1A1 (0.49) KDM4EALDH1A1L3MBTL1TDP1LMNA
SCHEMBL6606838 0.75 AGTR1 (0.53) KDM4EALDH1A1L3MBTL1TDP1LMNA
SCHEMBL9409377 0.75 AGTR1 (0.40) KDM4EALDH1A1HSD17B10
SCHEMBL6608915 0.74 AGTR1 (0.42) KDM4EALDH1A1L3MBTL1TDP1LMNA
SCHEMBL6606990 0.73 AGTR1 (0.57)
SCHEMBL8553595 0.71 LTB4R2 (0.45) KDM4EALDH1A1L3MBTL1TDP1LMNA
SCHEMBL2730 0.68 LTB4R2 (0.53) OXTRAVPR1ALTB4R2
SCHEMBL8550700 0.68 KDM4E (0.49) KDM4EALDH1A1L3MBTL1TDP1LMNA

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0588299-A2 1,2,4-Oxadiazolyl- or 1,2,4-thiadiazolyl-biphenyl derivatives as angiotensin II antagonists TAKEDA CHEMICAL INDUSTRIES, LTD. (JP) 1994-03-23 EP disclosed