SCHEMBL9409599

SCHEMBL9409599

COC(=O)CC[C@H]1CC[C@H](NC(=O)c2ccc(C3CCN(C(=O)OCOC(C)=O)CC3)cc2)CC1

nearest known ligand 0.44

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
HTR2A P28223 5/20 0.44
DRD3 P35462 5/20 0.44
DRD2 P14416 4/20 0.44
MAPT P10636 2/20 0.40
TSHR P16473 1/20 0.40
ALDH1A1 P00352 3/20 0.39
LMNA P02545 1/20 0.39
HDAC1 Q13547 1/20 0.38
TP53 P04637 1/20 0.38
HPGD P15428 1/20 0.38
CASP1 P29466 1/20 0.38
NPSR1 Q6W5P4 1/20 0.38
HSD17B10 Q99714 1/20 0.38
ENPP2 Q13822 1/20 0.38
PLG P00747 1/20 0.38
PRSS1 P07477 1/20 0.38
PRSS2 P07478 1/20 0.38
PRSS3 P35030 1/20 0.38
ST14 Q9Y5Y6 1/20 0.38
KDM4E B2RXH2 1/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9409396 0.90 HTR2A (0.49) HTR2ADRD3DRD2MAPTTSHR
SCHEMBL9409500 0.86 HDAC4 (0.48) HTR2ADRD3DRD2LMNAKDM4E
SCHEMBL9409398 0.83 HTR2A (0.52) HTR2ADRD3DRD2MAPTALDH1A1
SCHEMBL9409417 0.81 HRH3 (0.52) HTR2ADRD3DRD2MAPTALDH1A1
SCHEMBL9409541 0.81 PDE4B (0.46) HTR2ADRD3DRD2LMNAKDM4E
SCHEMBL9415854 0.78 ALDH1A1 (0.46) HTR2ADRD3DRD2MAPTALDH1A1
SCHEMBL9409367 0.78 ALDH1A1 (0.46) HTR2ADRD3DRD2MAPTALDH1A1
Hydrochloric Acid SCHEMBL9409523 0.78 ALDH1A1 (0.46) HTR2ADRD3DRD2MAPTALDH1A1
Hydrochloric Acid SCHEMBL9409352 0.78 ALDH1A1 (0.46) HTR2ADRD3DRD2MAPTALDH1A1
SCHEMBL4181896 0.74 HDAC4 (0.57) ALDH1A1LMNAKDM4E

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0604800-A1 4- 4- 4-(carboxyalkyl)-phenyl amino carbonyl -phenyl -piperedines as aggregation inhibitors Dr. Karl Thomae GmbH (DE) 1994-07-06 EP disclosed