Succinimide

Succinimide

SCHEMBL9417543

O=C(CBr)ON1C(=O)CCC1=O.O=C1CCC(=O)N1

nearest known ligand 0.38

Full drug profile on Sugi Atlas →

Predicted protein targets (top 5)

geneUniProtsupporting neighboursconfidence
CRBN Q96SW2 2/20 0.38
ADORA3 P0DMS8 1/20 0.31
ADORA2A P29274 1/20 0.31
ADORA2B P29275 1/20 0.31
MGLL Q99685 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL109446 0.89 TRPA1 (0.33) ADORA3ADORA2AADORA2BMGLL
SCHEMBL15624584 0.77
Succinimide SCHEMBL6549250 0.77 CRBN (0.42) CRBNMGLL
SCHEMBL15991602 0.76 TRPA1 (0.35)
SCHEMBL668588 0.75
SCHEMBL11125521 0.74 LMNA (0.34) MGLL
SCHEMBL3542603 0.74 KMT2A (0.35) MGLL
SCHEMBL28945733 0.74 MGLL (0.32) MGLL
SCHEMBL2568708 0.74 ADORA3 (0.37) ADORA3ADORA2AADORA2BMGLL
SCHEMBL2618714 0.73 MGLL (0.34) ADORA3ADORA2AADORA2BMGLL

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 7 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5373095-A Steroid compounds THE UPJOHN COMPANY (US) 1994-12-13 US disclosed
US-5334712-A Estrane or androstane pyridinyl alkyl or alkylphenyl amine steroids for antidiabetes and obesity THE UPJOHN COMPANY (US) 1994-08-02 US disclosed
US-5274089-A A estra-1,3,5(10)-triene derivative THE UPJOHN COMPANY (US) 1993-12-28 US disclosed
US-5196542-A Phospholipase A2 inhibitors THE UPJOHN COMPANY (US) 1993-03-23 US disclosed
US-5187299-A Phospholipase inhibitors; treating diabetes, obesity THE UPJOHN COMPANY (US) 1993-02-16 US disclosed
US-5145874-A Phospholipase inhibitor, hypoglycemic agent, antidiabetic, obesity THE UPJOHN COMPANY (US) 1992-09-08 US disclosed
US-4917826-A TREATING DIABETES AND OBESITY THE UPJOHN COMPANY (US) 1990-04-17 US disclosed