SCHEMBL9418976

SCHEMBL9418976

CC1CC(=O)CC(C)(C)c2ccc(Br)cc21

nearest known ligand 0.40

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 3/20 0.39
POLB P06746 1/20 0.39
TSHR P16473 1/20 0.39
HTR2A P28223 1/20 0.38
HTR2C P28335 1/20 0.38
HTR2B P41595 1/20 0.38
MEN1 O00255 1/20 0.37
KMT2A Q03164 1/20 0.37
OPRM1 P35372 2/20 0.37
OPRD1 P41143 2/20 0.37
OPRK1 P41145 2/20 0.37
CA1 P00915 1/20 0.36
CA2 P00918 1/20 0.36
PDE4B Q07343 1/20 0.35
CMA1 P23946 1/20 0.35
AHR P35869 1/20 0.35
BRD4 O60885 1/20 0.35
PBRM1 Q86U86 1/20 0.34
LMNA P02545 1/20 0.33
PKM P14618 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9418969 0.88 CMA1 (0.35) ALDH1A1POLBTSHRHTR2AHTR2C
SCHEMBL9418964 0.75 CMA1 (0.42) ALDH1A1KMT2APDE4BCMA1AHR
SCHEMBL18293057 0.74 HTR2B (0.41) ALDH1A1POLBTSHRHTR2AHTR2C
SCHEMBL8370875 0.71 TDP2 (0.47) ALDH1A1PDE4BCMA1AHRBRD4
SCHEMBL9419023 0.70 TDP2 (0.42) PDE4BCMA1AHRBRD4TDP2
SCHEMBL7796330 0.69 CMA1 (0.47) ALDH1A1PDE4BCMA1AHRBRD4
SCHEMBL9418949 0.68 CMA1 (0.42) ALDH1A1PDE4BCMA1AHRBRD4
SCHEMBL7928975 0.68 ADRA2A (0.40) HTR2AHTR2CHTR2BKMT2AOPRM1
SCHEMBL484599 0.67 PDE4B (0.46) MEN1KMT2ACA1CA2PDE4B
SCHEMBL4419838 0.67 PBRM1 (0.50) ALDH1A1POLBTSHRHTR2AHTR2C

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0315071-B1 Benzocyclohepten derivatives, their preparation and utilisation for pharmaceutics HOFFMANN LA ROCHE (CH) 1994-07-20 EP disclosed
US-4992574-A Skin disorders, antiallergens, antiinflammatory agent HOFFMANN-LA ROCHE INC. (US) 1991-02-12 US disclosed
EP-0315071-A2 Benzocyclohepten derivatives, their preparation and utilisation for pharmaceutics F. HOFFMANN-LA ROCHE AG (CH) 1989-05-10 EP disclosed