SCHEMBL9418969

SCHEMBL9418969

CC1CC(=O)CC(C)(C)c2cc(Br)ccc21

nearest known ligand 0.40

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CMA1 P23946 1/20 0.35
AHR P35869 1/20 0.35
HTR2A P28223 1/20 0.35
HTR2C P28335 1/20 0.35
HTR2B P41595 1/20 0.35
ALDH1A1 P00352 3/20 0.34
PBRM1 Q86U86 1/20 0.34
OPRM1 P35372 1/20 0.34
OPRD1 P41143 1/20 0.34
OPRK1 P41145 1/20 0.34
LMNA P02545 1/20 0.33
PKM P14618 1/20 0.33
TDP2 O95551 1/20 0.33
CA1 P00915 1/20 0.33
CA2 P00918 1/20 0.33
POLB P06746 1/20 0.33
TSHR P16473 1/20 0.33
ADRA2A P08913 1/20 0.33
PNMT P11086 1/20 0.33
ADRA2B P18089 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9418976 0.88 ALDH1A1 (0.39) CMA1AHRHTR2AHTR2CHTR2B
SCHEMBL9418964 0.75 CMA1 (0.42) CMA1AHRALDH1A1TDP2KMT2A
SCHEMBL7796330 0.72 CMA1 (0.47) CMA1AHRALDH1A1TDP2
SCHEMBL9418949 0.71 CMA1 (0.42) CMA1AHRALDH1A1TDP2
SCHEMBL7928975 0.71 ADRA2A (0.40) CMA1AHRHTR2AHTR2CHTR2B
SCHEMBL8370875 0.68 TDP2 (0.47) CMA1AHRALDH1A1TDP2ADRA2A
SCHEMBL3361527 0.67 PGR (0.55) CMA1AHRHTR2AHTR2CALDH1A1
SCHEMBL14169119 0.67 PBRM1 (0.54) HTR2AHTR2CHTR2BPBRM1OPRM1
SCHEMBL26656332 0.67 PBRM1 (0.54) HTR2AHTR2CHTR2BPBRM1OPRM1
SCHEMBL9419023 0.67 TDP2 (0.42) CMA1AHRTDP2PNMT

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0315071-B1 Benzocyclohepten derivatives, their preparation and utilisation for pharmaceutics HOFFMANN LA ROCHE (CH) 1994-07-20 EP disclosed
US-4992574-A Skin disorders, antiallergens, antiinflammatory agent HOFFMANN-LA ROCHE INC. (US) 1991-02-12 US disclosed