SCHEMBL9419643

SCHEMBL9419643

O=C(CN1CCNCC1CCO)N1c2ccccc2Oc2ccccc21

nearest known ligand 0.42

Predicted protein targets (top 11)

geneUniProtsupporting neighboursconfidence
CA1 P00915 2/20 0.40
CA2 P00918 2/20 0.40
CA4 P22748 2/20 0.40
CA9 Q16790 2/20 0.40
P2RX4 Q99571 12/20 0.39
ALDH1A1 P00352 1/20 0.35
ALOX15 P16050 1/20 0.35
P2RX1 P51575 2/20 0.35
P2RX3 P56373 1/20 0.35
CACNA1H O95180 1/20 0.35
CACNA1B Q00975 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6045358 0.91 PIM1 (0.43) P2RX4ALDH1A1ALOX15
SCHEMBL6045244 0.79 PIM1 (0.41) CA1CA2CA4CA9
SCHEMBL11817278 0.72 CHRM2 (0.53)
SCHEMBL6045312 0.72 PIM1 (0.56) ALDH1A1CACNA1B
SCHEMBL6045308 0.72 PIM1 (0.56) ALDH1A1CACNA1B
SCHEMBL23496876 0.69 SIGMAR1 (0.54) CA1CA2CA4CA9ALDH1A1
SCHEMBL6008090 0.69 SIGMAR1 (0.54) CA1CA2CA4CA9ALDH1A1
SCHEMBL3948948 0.69 SIGMAR1 (0.54) CA1CA2CA4CA9ALDH1A1
SCHEMBL9419617 0.69 ALDH1A1 (0.64) P2RX4ALDH1A1ALOX15CACNA1HCACNA1B
SCHEMBL9419641 0.68 ALDH1A1 (0.62) P2RX4ALDH1A1ALOX15CACNA1HCACNA1B

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5371081-A Useful in potentiating the cytotoxic effect of chemotherapeutic agents ST. JUDE CHILDREN'S RESEARCH HOSPITAL (US) 1994-12-06 US claimed
WO-1993003729-A1 N-SUBSTITUTED PHENOXAZINES FOR TREATING MULTIDRUG RESISTANT CANCER CELLS RESEARCH CORPORATION TECHNOLOGIES, INC. (US) 1993-03-04 WO claimed
US-5371081-A Useful in potentiating the cytotoxic effect of chemotherapeutic agents ST. JUDE CHILDREN'S RESEARCH HOSPITAL (US) 1994-12-06 US disclosed
WO-1993003729-A1 N-SUBSTITUTED PHENOXAZINES FOR TREATING MULTIDRUG RESISTANT CANCER CELLS RESEARCH CORPORATION TECHNOLOGIES, INC. (US) 1993-03-04 WO disclosed