SCHEMBL9428162

SCHEMBL9428162

Cn1c(N2CCN(CCOc3ccccc3N)CC2)cc(=O)n(C)c1=O

nearest known ligand 0.47

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
LTA4H P09960 1/20 0.47
MEN1 O00255 1/20 0.47
ALDH1A1 P00352 1/20 0.47
KMT2A Q03164 1/20 0.47
HRH1 P35367 7/20 0.44
HTR1A P08908 5/20 0.44
ADRA1A P35348 4/20 0.44
DRD2 P14416 3/20 0.44
MAPT P10636 2/20 0.44
ADRA2A P08913 2/20 0.44
ADRA2B P18089 2/20 0.44
ADRA2C P18825 2/20 0.44
DRD3 P35462 2/20 0.44
HTR2B P41595 2/20 0.44
CYP2C19 P33261 2/20 0.44
LMNA P02545 1/20 0.44
ADRB2 P07550 1/20 0.44
ADRB1 P08588 1/20 0.44
CYP3A4 P08684 1/20 0.44
CYP2C9 P11712 1/20 0.44

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9428336 0.94 HRH1 (0.48) MEN1ALDH1A1KMT2AHRH1HTR1A
SCHEMBL9429100 0.93 HRH1 (0.49) MEN1ALDH1A1KMT2AHRH1HTR1A
Oxalic Acid SCHEMBL9430076 0.89 ALDH1A1 (0.49) MEN1ALDH1A1KMT2AHRH1HTR1A
SCHEMBL9429366 0.84 ALDH1A1 (0.52) LTA4HMEN1ALDH1A1KMT2AHRH1
SCHEMBL9429465 0.83 MAPT (0.52) MEN1ALDH1A1KMT2AHRH1HTR1A
Hydrochloric Acid SCHEMBL9428580 0.83 MEN1 (0.51) LTA4HMEN1ALDH1A1KMT2AHRH1
SCHEMBL9428616 0.82 DRD2 (0.44) MEN1ALDH1A1KMT2AHRH1HTR1A
SCHEMBL9429697 0.81 DRD2 (0.57) ALDH1A1HRH1HTR1AADRA1ADRD2
SCHEMBL9429282 0.81 KDM4E (0.54) MEN1ALDH1A1KMT2AHRH1HTR1A
SCHEMBL9429005 0.81 CYP2C19 (0.53) MEN1ALDH1A1KMT2AHRH1HTR1A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5332739-A Pyrimidinedione derivatives and antiarrhythmic agents containing same MITSUI TOATSU CHEMICALS, INCORPORATED (JP) 1994-07-26 US disclosed
EP-0454498-A2 Pyrimidinedione derivatives and antiarrhythmic agents containing same MITSUI TOATSU CHEMICALS, Inc. (JP) 1991-10-30 EP disclosed