SCHEMBL9428804

SCHEMBL9428804

COc1ccc(CCN2CCN(c3cc(=O)n(C)c(=O)n3C)CC2)cc1F

nearest known ligand 0.50

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 2/20 0.45
MEN1 O00255 1/20 0.45
KMT2A Q03164 1/20 0.45
HTR1A P08908 3/20 0.45
HTR2C P28335 2/20 0.45
ADRA1B P35368 3/20 0.44
ADRA1A P35348 3/20 0.44
ADRA1D P25100 2/20 0.44
EBP Q15125 2/20 0.44
SIGMAR1 Q99720 2/20 0.44
TMEM97 Q5BJF2 1/20 0.44
HRH1 P35367 2/20 0.43
MAPT P10636 2/20 0.43
LMNA P02545 1/20 0.43
ADRB2 P07550 1/20 0.43
ADRB1 P08588 1/20 0.43
CYP3A4 P08684 1/20 0.43
ADRA2A P08913 1/20 0.43
CYP2C9 P11712 1/20 0.43
DRD2 P14416 1/20 0.43

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9385849 0.81 HTR1A (0.51) ALDH1A1MEN1KMT2AHTR1AHRH1
SCHEMBL9428322 0.79 SLC6A3 (0.57) ALDH1A1MEN1KMT2AHTR1ASIGMAR1
SCHEMBL9428318 0.78 MEN1 (0.54) ALDH1A1MEN1KMT2AADRA1BADRA1A
SCHEMBL9428246 0.77 MEN1 (0.52) ALDH1A1MEN1KMT2AHTR1AADRA1B
SCHEMBL9428716 0.77 ALDH1A1 (0.52) ALDH1A1MEN1KMT2AHTR1AADRA1B
SCHEMBL9429643 0.77 MEN1 (0.55) ALDH1A1MEN1KMT2AHTR1AADRA1B
Hydrochloric Acid SCHEMBL9428320 0.76 MEN1 (0.51) ALDH1A1MEN1KMT2AHTR1AADRA1B
Hydrochloric Acid SCHEMBL9428451 0.76 MEN1 (0.54) ALDH1A1MEN1KMT2AHTR1AADRA1B
SCHEMBL9428993 0.75 ALDH1A1 (0.50) ALDH1A1MEN1KMT2AADRA1BADRA1A
SCHEMBL5183284 0.74 SIGMAR1 (0.47) ADRA1BADRA1AADRA1DEBPSIGMAR1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5332739-A Pyrimidinedione derivatives and antiarrhythmic agents containing same MITSUI TOATSU CHEMICALS, INCORPORATED (JP) 1994-07-26 US disclosed
EP-0454498-A2 Pyrimidinedione derivatives and antiarrhythmic agents containing same MITSUI TOATSU CHEMICALS, Inc. (JP) 1991-10-30 EP disclosed