SCHEMBL9433558

SCHEMBL9433558

O=C(C=Cc1ccccc1C(F)(F)F)Cc1cccnc1

nearest known ligand 0.54

Predicted protein targets (top 16)

geneUniProtsupporting neighboursconfidence
NFKB1 P19838 1/20 0.54
BACE1 P56817 1/20 0.52
MAOB P27338 8/20 0.47
NFE2L2 Q16236 2/20 0.46
P4HB P07237 1/20 0.46
ABCG2 Q9UNQ0 1/20 0.46
NAPRT Q6XQN6 1/20 0.46
CYP1A2 P05177 1/20 0.45
CYP3A4 P08684 1/20 0.45
CYP2C9 P11712 1/20 0.45
MAOA P21397 1/20 0.43
FDPS P14324 1/20 0.43
LMNA P02545 2/20 0.43
MEN1 O00255 1/20 0.43
MAPT P10636 1/20 0.43
KMT2A Q03164 1/20 0.43

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9434718 0.82 NAPRT (0.50) NFKB1NFE2L2NAPRTCYP1A2CYP3A4
SCHEMBL9433617 0.81 HSD11B1 (0.50) NAPRTCYP1A2CYP3A4CYP2C9LMNA
SCHEMBL9433799 0.81 MAPT (0.61) MAOBNAPRTCYP1A2CYP3A4CYP2C9
SCHEMBL9434498 0.81 NAPRT (0.49) NAPRTCYP1A2CYP3A4CYP2C9LMNA
SCHEMBL9433573 0.81 NAPRT (0.49) NAPRTCYP1A2CYP3A4CYP2C9LMNA
SCHEMBL9434607 0.79 CYP1A2 (0.53) BACE1NAPRTCYP1A2CYP3A4CYP2C9
SCHEMBL9433343 0.79 TBXAS1 (0.52) MAOBP4HBNAPRTCYP1A2CYP3A4
SCHEMBL9433528 0.78 NAPRT (0.46) NAPRTCYP1A2CYP3A4CYP2C9LMNA
SCHEMBL9433587 0.77 ALDH1A1 (0.61) NFKB1BACE1MAOBLMNAMEN1
SCHEMBL9434583 0.76 KMT2A (0.49) NAPRTCYP1A2CYP3A4CYP2C9LMNA

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5276150-A Vasodilators, anticoagulants, calcium channel blockers FUJIREBIO INC. (JP) 1994-01-04 US disclosed
EP-0400660-A1 1,4-dihydropyridine derivatives FUJIREBIO INC. (JP) 1990-12-05 EP disclosed