SCHEMBL9433711

SCHEMBL9433711

C=CC(=O)Cc1cnccc1-c1cccc2cnccc12

nearest known ligand 0.44

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
SLC22A12 Q96S37 2/20 0.44
KDM4E B2RXH2 1/20 0.41
MAPKAPK2 P49137 1/20 0.41
IKBKE Q14164 1/20 0.40
TBK1 Q9UHD2 1/20 0.40
ROS1 P08922 1/20 0.40
RPS6KB1 P23443 1/20 0.40
GLS O94925 1/20 0.39
HTT P42858 1/20 0.38
LMNA P02545 1/20 0.38
CYP1A2 P05177 1/20 0.38
CYP3A4 P08684 1/20 0.38
CYP2D6 P10635 1/20 0.38
CYP2C9 P11712 1/20 0.38
CYP2C19 P33261 1/20 0.38
CCNE1 P24864 1/20 0.38
CDK2 P24941 1/20 0.38
CDK5 Q00535 1/20 0.38
MAPK8 P45983 5/20 0.37
MAPK9 P45984 5/20 0.37

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9434522 0.92 SLC22A12 (0.44) SLC22A12IKBKETBK1ROS1RPS6KB1
SCHEMBL9434508 0.80 GPBAR1 (0.43)
SCHEMBL9434729 0.80 MAOA (0.36) KDM4ELMNACYP3A4CDK5KCNA5
SCHEMBL9434595 0.80 MEN1 (0.38) KDM4EKCNA5
SCHEMBL9433586 0.79 MAOA (0.35) CYP1A2CYP2D6CYP2C9CYP2C19KCNA5
SCHEMBL9433807 0.79 LIMK1 (0.41)
SCHEMBL9433625 0.79 KMT2A (0.35) KDM4EGLSKCNA5
SCHEMBL9433611 0.77 ALDH1A1 (0.36) SLC22A12KDM4EHTTCYP1A2CYP3A4
SCHEMBL9433930 0.76 GPBAR1 (0.36) SLC22A12CYP1A2CYP3A4CYP2D6CYP2C9
SCHEMBL9434105 0.76 RECQL (0.36) KDM4ECYP1A2CYP3A4CYP2C19

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5276150-A Vasodilators, anticoagulants, calcium channel blockers FUJIREBIO INC. (JP) 1994-01-04 US disclosed
EP-0400660-A1 1,4-dihydropyridine derivatives FUJIREBIO INC. (JP) 1990-12-05 EP disclosed