SCHEMBL9434729

SCHEMBL9434729

C=CC(=O)Cc1cnccc1-c1ccccc1O

nearest known ligand 0.36

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
MAOA P21397 1/20 0.36
MAOB P27338 1/20 0.36
GSTO1 P78417 1/20 0.35
HPGD P15428 1/20 0.34
RAB9A P51151 1/20 0.34
L3MBTL1 Q9Y468 1/20 0.34
CCNC P24863 1/20 0.33
CDK8 P49336 1/20 0.33
HASPIN Q8TF76 1/20 0.33
IDO1 P14902 1/20 0.33
AKR1B1 P15121 1/20 0.33
ROCK1 Q13464 1/20 0.33
KDM4E B2RXH2 1/20 0.33
KCNA5 P22460 1/20 0.32
ROCK2 O75116 1/20 0.32
CCNB2 O95067 1/20 0.32
CDK1 P06493 1/20 0.32
CCNB1 P14635 1/20 0.32
GSK3A P49840 1/20 0.32
GSK3B P49841 1/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9434508 0.86 GPBAR1 (0.43) GPBAR1
SCHEMBL9433586 0.85 MAOA (0.35) MAOAMAOBKCNA5GPBAR1
SCHEMBL9433625 0.85 KMT2A (0.35) MAOAMAOBHPGDRAB9ACCNC
SCHEMBL9433807 0.85 LIMK1 (0.41) GSTO1GSK3AGSK3BGPBAR1
SCHEMBL9434522 0.83 SLC22A12 (0.44) HPGDKCNA5MAPTSMN1; SMN2CYP3A4
SCHEMBL9433534 0.82 GPBAR1 (0.42) HPGDGPBAR1CYP3A4
SCHEMBL9433598 0.81 RORC (0.40) RAB9AL3MBTL1KDM4ELMNAMAPT
SCHEMBL9434595 0.80 MEN1 (0.38) KDM4EKCNA5ROCK2
SCHEMBL9433711 0.80 SLC22A12 (0.44) KDM4EKCNA5CDK5LMNACYP3A4
SCHEMBL9433930 0.80 GPBAR1 (0.36) HPGDCCNCCDK8KCNA5GSK3A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5276150-A Vasodilators, anticoagulants, calcium channel blockers FUJIREBIO INC. (JP) 1994-01-04 US disclosed
EP-0400660-A1 1,4-dihydropyridine derivatives FUJIREBIO INC. (JP) 1990-12-05 EP disclosed