SCHEMBL9433742

SCHEMBL9433742

CC(C)Oc1oc(C(N)=O)c2ccc(-c3ccccc3)cc12

nearest known ligand 0.43

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
RXRA P19793 1/20 0.43
RXRB P28702 1/20 0.43
MEN1 O00255 2/20 0.41
MAPT P10636 2/20 0.41
KMT2A Q03164 2/20 0.41
SMN1; SMN2 Q16637 2/20 0.41
LMNA P02545 1/20 0.41
TP53 P04637 1/20 0.41
CYP3A4 P08684 1/20 0.41
LRRK2 Q5S007 2/20 0.40
MKNK1 Q9BUB5 1/20 0.39
MKNK2 Q9HBH9 1/20 0.39
IRAK4 Q9NWZ3 2/20 0.38
GAA P10253 2/20 0.38
CYP1A2 P05177 1/20 0.38
CYP2C9 P11712 1/20 0.38
PKM P14618 1/20 0.38
CYP2C19 P33261 1/20 0.38
PDCD1 Q15116 1/20 0.38
CD274 Q9NZQ7 1/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9432939 0.90 RXRA (0.48) RXRARXRBMEN1MAPTKMT2A
SCHEMBL27280518 0.86 NR4A2 (0.44) RXRARXRBMEN1MAPTKMT2A
SCHEMBL9433908 0.83 IRAK4 (0.46) MEN1MAPTKMT2ASMN1; SMN2LMNA
SCHEMBL9432880 0.80 KDM4E (0.47) SMN1; SMN2LMNAIRAK4GAAALDH1A1
SCHEMBL9433688 0.79 ICAM1 (0.51) MEN1MAPTKMT2ASMN1; SMN2LMNA
SCHEMBL9433079 0.79 EDNRA (0.51) PKMNPC1CASP3RAB9ASENP8
SCHEMBL9433730 0.79 KDM4E (0.43) RXRARXRBMEN1MAPTKMT2A
SCHEMBL10375126 0.76 ADCY1 (0.37) RXRARXRBMEN1MAPTKMT2A
SCHEMBL10374754 0.74 NR4A2 (0.41) ALDH1A1BRD4HPGDKDM4E
SCHEMBL9434171 0.73 KMT2A (0.40) RXRARXRBMEN1MAPTKMT2A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5350748-A 3-thio or amino substituted-benzo[b]thiophene-2-carboxamides and 3-oxygen, thio, or amino substituted-benzofuran-2-carboxamides as inhibitors of cell adhesion WARNER-LAMBERT COMPANY (US) 1994-09-27 US disclosed