SCHEMBL9433919

SCHEMBL9433919

CC1=C(C(=O)O)C(c2ccc(Br)cc2)C(c2cccnc2)=C(C)N1

nearest known ligand 0.44

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CACNA1B Q00975 1/20 0.44
KMT2A Q03164 2/20 0.41
RXFP1 Q9HBX9 2/20 0.41
ALDH1A1 P00352 8/20 0.39
KDM4E B2RXH2 7/20 0.39
GAA P10253 6/20 0.39
HPGD P15428 5/20 0.39
CASP1 P29466 3/20 0.39
CASP7 P55210 3/20 0.39
HSD17B10 Q99714 3/20 0.39
FFAR3 O14843 1/20 0.38
ABL1 P00519 1/20 0.38
LMNA P02545 1/20 0.38
RIN1 Q13671 1/20 0.38
MKNK1 Q9BUB5 1/20 0.38
MKNK2 Q9HBH9 1/20 0.38
MAPT P10636 2/20 0.38
NPSR1 Q6W5P4 2/20 0.38
GLA P06280 2/20 0.38
POLB P06746 1/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9434755 0.91 CACNA1B (0.45) CACNA1BKMT2AALDH1A1KDM4EGAA
SCHEMBL10432705 0.89 CACNA1B (0.44) CACNA1BALDH1A1KDM4EGAAHPGD
SCHEMBL9434417 0.88 MAPT (0.45) CACNA1BKMT2AALDH1A1KDM4EGAA
SCHEMBL9434316 0.88 CACNA1B (0.44) CACNA1BALDH1A1KDM4EGAAHPGD
SCHEMBL9433827 0.88 CACNA1B (0.48) CACNA1BKMT2ARXFP1ALDH1A1KDM4E
SCHEMBL10432690 0.88 HSD17B10 (0.48) KMT2AALDH1A1KDM4EGAAHPGD
SCHEMBL9434041 0.86 CACNA1B (0.42) CACNA1BKMT2AALDH1A1KDM4EGAA
SCHEMBL9433821 0.86 ALDH1A1 (0.46) CACNA1BKMT2AALDH1A1KDM4EGAA
SCHEMBL9433669 0.83 ALDH1A1 (0.47) CACNA1BKMT2AALDH1A1KDM4EGAA
SCHEMBL9434792 0.83 CACNA1B (0.43) CACNA1BALDH1A1GAAMKNK1MKNK2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5276150-A Vasodilators, anticoagulants, calcium channel blockers FUJIREBIO INC. (JP) 1994-01-04 US disclosed
EP-0400660-A1 1,4-dihydropyridine derivatives FUJIREBIO INC. (JP) 1990-12-05 EP disclosed