SCHEMBL9434755

SCHEMBL9434755

CC1=C(C(=O)O)C(c2ccc(C)cc2)C(c2cccnc2)=C(C)N1

nearest known ligand 0.45

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CACNA1B Q00975 1/20 0.45
ALDH1A1 P00352 9/20 0.40
KDM4E B2RXH2 7/20 0.40
GAA P10253 6/20 0.40
HPGD P15428 5/20 0.40
CASP1 P29466 3/20 0.40
CASP7 P55210 3/20 0.40
HSD17B10 Q99714 3/20 0.40
MAPT P10636 2/20 0.40
F2 P00734 1/20 0.40
KLK7 P49862 1/20 0.40
KMT2A Q03164 1/20 0.40
KLK14 Q9P0G3 1/20 0.40
KLK5 Q9Y337 1/20 0.40
ST14 Q9Y5Y6 1/20 0.40
MKNK1 Q9BUB5 1/20 0.40
MKNK2 Q9HBH9 1/20 0.40
CYP3A4 P08684 1/20 0.40
CYP2A6 P11509 1/20 0.40
SMN1; SMN2 Q16637 2/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL10432705 0.92 CACNA1B (0.44) CACNA1BALDH1A1KDM4EGAAHPGD
SCHEMBL9433919 0.91 CACNA1B (0.44) CACNA1BALDH1A1KDM4EGAAHPGD
SCHEMBL9434417 0.91 MAPT (0.45) CACNA1BALDH1A1KDM4EGAAHPGD
SCHEMBL9434316 0.91 CACNA1B (0.44) CACNA1BALDH1A1KDM4EGAAHPGD
SCHEMBL9433821 0.89 ALDH1A1 (0.46) CACNA1BALDH1A1KDM4EGAAHPGD
SCHEMBL9434041 0.89 CACNA1B (0.42) CACNA1BALDH1A1KDM4EGAAHPGD
SCHEMBL9434335 0.87 TSHR (0.48) ALDH1A1KDM4EGAAHPGDCASP1
SCHEMBL9433669 0.87 ALDH1A1 (0.47) CACNA1BALDH1A1KDM4EGAAHPGD
SCHEMBL9434087 0.85 CACNA1B (0.43) CACNA1BALDH1A1KDM4EGAAHPGD
SCHEMBL7277208 0.85 MKNK1 (0.54) CACNA1BMAPTKMT2AMKNK1MKNK2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5276150-A Vasodilators, anticoagulants, calcium channel blockers FUJIREBIO INC. (JP) 1994-01-04 US disclosed
EP-0400660-A1 1,4-dihydropyridine derivatives FUJIREBIO INC. (JP) 1990-12-05 EP disclosed