SCHEMBL8997253

SCHEMBL8997253

CCC(CCC1CNc2nc(N)nc(N)c21)c1ccc(C(=O)N[C@@H](CCC(=O)O)C(=O)O)cc1

nearest known ligand 0.70

Predicted protein targets (top 3)

geneUniProtsupporting neighboursconfidence
DHFR P00374 2/20 0.58
ATIC P31939 2/20 0.52
GART P22102 3/20 0.49

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9397716 0.94 DHFR (0.53) DHFRATICGART
SCHEMBL8997170 0.90 DHFR (0.55) DHFRATICGART
SCHEMBL9758306 0.90 DHFR (0.55) DHFRATICGART
SCHEMBL9758337 0.90 DHFR (0.60) DHFRATICGART
SCHEMBL8997198 0.90 ATIC (0.48) DHFRATICGART
SCHEMBL9227822 0.87 DHFR (0.52) DHFRATICGART
SCHEMBL8997146 0.86 ATIC (0.50) DHFRATICGART
SCHEMBL8997214 0.86 ATIC (0.49) ATICGART
SCHEMBL9439698 0.85 GART (0.48) DHFRATICGART
SCHEMBL9088274 0.84 ATIC (0.51) DHFRATICGART

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 9 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0334636-B1 Pyrrolopyrimidine derivatives, their production and use TAKEDA CHEMICAL INDUSTRIES LTD (JP) 1996-10-23 EP disclosed
US-5539113-A ANTITUMOR AGENTS TAKEDA CHEMICAL INDUSTRIES, LTD. (JP) 1996-07-23 US disclosed
US-5496946-A Production of pyrrolopyrimidines and intermediates therefor TAKEDA CHEMICAL INDUSTRIES, LTD. (JP) 1996-03-05 US disclosed
US-5349064-A Production of pyrrolopyrimidines TAKEDA CHEMICAL INDUSTRIES, LTD. (JP) 1994-09-20 US disclosed
US-5296600-A Antitumor agents TAKEDA CHEMICAL INDUSTRIES, LTD. (JP) 1994-03-22 US disclosed
US-5106974-A Antitumor and -carcinogenic agents TAKEDA CHEMICAL INDUSTRIES, LTD. (JP) 1992-04-21 US disclosed
US-4997838-A Antitumor agents TAKEDA CHEMICAL INDUSTRIES, LTD. (JP) 1991-03-05 US disclosed
EP-0402903-A1 Production of pyrrolopyrimidines and intermediates therefor Takeda Chemical Industries, Ltd. (JP) 1990-12-19 EP disclosed
EP-0334636-A2 Pyrrolopyrimidine derivatives, their production and use Takeda Chemical Industries, Ltd. (JP) 1989-09-27 EP disclosed