SCHEMBL9440949

SCHEMBL9440949

CN(C(=O)O)c1ncc[nH]1

nearest known ligand 0.39

Predicted protein targets (top 18)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 4/20 0.37
KDM4E B2RXH2 3/20 0.37
SMN1; SMN2 Q16637 1/20 0.37
RAB9A P51151 2/20 0.36
NPC1 O15118 1/20 0.36
TBXAS1 P24557 2/20 0.35
TAAR1 Q96RJ0 2/20 0.35
ADRA2A P08913 1/20 0.34
ADRA2B P18089 1/20 0.34
ADRA2C P18825 1/20 0.34
HTR1A P08908 1/20 0.32
MTOR P42345 1/20 0.31
ADK P55263 1/20 0.31
NISCH Q9Y2I1 1/20 0.31
CYP3A4 P08684 1/20 0.31
TSHR P16473 1/20 0.31
CYP2C19 P33261 1/20 0.31
LMNA P02545 1/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL391774 0.84 ALDH1A1 (0.37) ALDH1A1KDM4ESMN1; SMN2RAB9ANPC1
SCHEMBL31169778 0.79 ALDH1A1 (0.39) ALDH1A1KDM4ESMN1; SMN2RAB9ANPC1
SCHEMBL4564864 0.79 KDM4E (0.49) ALDH1A1KDM4ESMN1; SMN2RAB9ANPC1
SCHEMBL10612608 0.78 NPC1 (0.33) ALDH1A1KDM4ESMN1; SMN2RAB9ANPC1
SCHEMBL7426536 0.77 TAAR1 (0.38) ALDH1A1KDM4ESMN1; SMN2RAB9ANPC1
SCHEMBL29003727 0.77 FFAR2 (0.42) ALDH1A1KDM4EADRA2AADRA2C
SCHEMBL2837058 0.76 TAAR1 (0.42) ALDH1A1KDM4ESMN1; SMN2RAB9ANPC1
SCHEMBL3684538 0.76 ALDH1A1 (0.38) ALDH1A1KDM4ESMN1; SMN2RAB9ANPC1
SCHEMBL1853863 0.75 LMNA (0.38) ALDH1A1KDM4ESMN1; SMN2RAB9ANPC1
SCHEMBL2424191 0.75 PAX8 (0.35) ALDH1A1KDM4ESMN1; SMN2RAB9ANPC1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 19 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-3220910-A1 AMINOPYRAZINE COMPOUNDS WITH A2A ANTAGONIST PROPERTIES Merck Sharp & Dohme Corp. (US) 2017-09-27 EP disclosed
WO-2016081290-A1 AMINOPYRAZINE COMPOUNDS WITH A2A ANTAGONIST PROPERTIES MERCK SHARP & DOHME CORP. (US) 2016-05-26 WO disclosed
WO-2012088124-A2 TETRAHYDRO-AZACARBOLINE MCH-1 ANTAGONISTS, METHODS OF MAKING, AND USES THEREOF ALBANY MOLECULAR RESEARCH, INC. (US) 2012-06-28 WO disclosed
EP-0244177-B1 Method for processing light-sensitive silver halide color photographic material KONISHIROKU PHOTO IND (JP) 1994-05-04 EP disclosed
EP-0296854-B1 METHOD FOR PROCESSING LIGHT-SENSITIVE SILVER HALIDE COLOR PHOTOGRAPHIC MATERIAL KONICA CORPORATION (JP) 1993-08-18 EP disclosed
EP-0168263-B1 METHOD FOR PROCESSING LIGHT-SENSITIVE SILVER HALIDE PHOTOGRAPHIC MATERIAL KONICA CORPORATION (JP) 1991-04-10 EP disclosed
EP-0217643-B1 METHOD FOR PROCESSING LIGHT-SENSITIVE SILVER HALIDE COLOR PHOTOGRAPHIC MATERIAL KONICA CORPORATION (JP) 1991-01-23 EP disclosed
US-4983503-A BLEACH-FIXING KONICA CORPORATION (JP) 1991-01-08 US disclosed
EP-0199604-B1 PROCESSING METHOD FOR LIGHT-SENSITIVE SILVER HALIDE COLOR PHOTOGRAPHIC MATERIAL KONICA CORPORATION (JP) 1990-12-27 EP disclosed
US-4914008-A Bleach fixing after color development KONISHIROKU PHOTO INDUSTRY CO., LTD. (JP) 1990-04-03 US disclosed
EP-0337560-A2 2-Phenylsulfinyl-nitro-pyridines, process for their preparation and their use BAYER AG (DE) 1989-10-18 EP disclosed
EP-0336186-A2 Derivatives of triazolylmethylcyclopropyl-carbinols as material protecting agents BAYER AG (DE) 1989-10-11 EP disclosed
EP-0298338-A1 Microbicidal agents BAYER AG (DE) 1989-01-11 EP disclosed
EP-0296854-A2 Method for processing light-sensitive silver halide color photographic material KONICA CORPORATION (JP) 1988-12-28 EP disclosed
US-4778743-A ALDEHYDE DERIVATIVE KONISHIROKU PHOTO INDUSTRY CO., LTD. (JP) 1988-10-18 US disclosed
US-4778748-A Method for processing light-sensitive silver halide color photographic material KONISHIROKU PHOTO INDUSTRIES, CO., LTD. (JP) 1988-10-18 US disclosed
EP-0244177-A2 Method for processing light-sensitive silver halide color photographic material KONICA CORPORATION (JP) 1987-11-04 EP disclosed
EP-0217643-A2 Method for processing light-sensitive silver halide color photographic material KONICA CORPORATION (JP) 1987-04-08 EP disclosed
EP-0199604-A2 Processing method for light-sensitive silver halide color photographic material KONICA CORPORATION (JP) 1986-10-29 EP disclosed