SCHEMBL9444479

SCHEMBL9444479

COc1cc(NS(C)(=O)=O)ccc1C(=O)C1CCN(C(C)=O)CC1

nearest known ligand 0.43

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
HSD11B1 P28845 1/20 0.43
CPS1 P31327 1/20 0.42
QDPR P09417 1/20 0.42
SMN1; SMN2 Q16637 3/20 0.41
L3MBTL1 Q9Y468 1/20 0.41
CYP17A1 P05093 1/20 0.41
ACHE P22303 1/20 0.41
BACE1 P56817 1/20 0.41
ALDH1A1 P00352 2/20 0.41
KDM2B Q8NHM5 3/20 0.40
GLA P06280 2/20 0.40
REV1 Q9UBZ9 1/20 0.40
SLC22A1 O15245 1/20 0.40
ABCC4 O15439 1/20 0.40
KDM1A O60341 1/20 0.40
NR1I2 O75469 1/20 0.40
TP53 P04637 1/20 0.40
CYP1A2 P05177 1/20 0.40
CYP3A4 P08684 1/20 0.40
CYP2D6 P10635 1/20 0.40

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9444485 0.85 SMN1; SMN2 (0.43) CPS1QDPRSMN1; SMN2ALDH1A1REV1
Hydrochloric Acid SCHEMBL9444506 0.83 KDM1A (0.47) SMN1; SMN2CYP17A1ALDH1A1KDM2BGLA
SCHEMBL9444322 0.80 ACHE (0.47) CYP17A1ACHEALDH1A1KDM4EKMT2A
SCHEMBL6712581 0.80 HSD11B1 (0.63) HSD11B1CPS1SMN1; SMN2L3MBTL1ALDH1A1
SCHEMBL9444360 0.78 KCNH2 (0.57) HSD11B1L3MBTL1TP53CYP1A2CYP3A4
SCHEMBL6281251 0.74 TSHR (0.45) HSD11B1CPS1SMN1; SMN2L3MBTL1ACHE
SCHEMBL5359155 0.74 ALDH1A1 (0.53) SMN1; SMN2CYP17A1ALDH1A1GLASLC22A1
SCHEMBL23215646 0.73 MGLL (0.49) HSD11B1CPS1QDPRSMN1; SMN2ALDH1A1
SCHEMBL29745184 0.73 MGLL (0.49) HSD11B1CPS1QDPRSMN1; SMN2ALDH1A1
SCHEMBL12970664 0.73 MEN1 (0.52) SMN1; SMN2CYP17A1ALDH1A1GLASLC22A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 6 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0235752-B1 Piperidine derivative, pharmaceutical composition containing the same and use EISAI CO LTD (JP) 1993-11-18 EP disclosed
US-5179095-A Antiarrhythmia agents EISAI CO., LTD. (JP) 1993-01-12 US disclosed
US-5118689-A Antiarrhythmia agents EISAI CO., LTD. (JP) 1992-06-02 US disclosed
US-4996215-A Antiarrythmia agents EISAI CO., LTD. (JP) 1991-02-26 US disclosed
US-4876262-A ANTIARRHYTHMIA AGENTS EISAI CO., LTD. (JP) 1989-10-24 US disclosed
EP-0235752-A2 Piperidine derivative, pharmaceutical composition containing the same and use Eisai Co., Ltd. (JP) 1987-09-09 EP disclosed