SCHEMBL9448951

SCHEMBL9448951

[N-]=[N+]=CC(=O)c1ccccc1Br

nearest known ligand 0.46

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 6/20 0.46
LMNA P02545 2/20 0.46
TP53 P04637 1/20 0.46
HSP90AA1 P07900 1/20 0.42
MAPT P10636 1/20 0.42
ATM Q13315 1/20 0.42
NPSR1 Q6W5P4 1/20 0.42
MEN1 O00255 4/20 0.41
KMT2A Q03164 4/20 0.41
HTT P42858 1/20 0.41
HIF1A Q16665 1/20 0.41
MAOB P27338 1/20 0.40
NPC1 O15118 1/20 0.40
RAB9A P51151 1/20 0.40
HPGD P15428 2/20 0.39
ELANE P08246 1/20 0.38
POLB P06746 2/20 0.37
CYP1A2 P05177 1/20 0.37
CYP2C9 P11712 1/20 0.37
CYP2C19 P33261 1/20 0.37

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL204224 0.79 PRNP (0.41) ALDH1A1LMNAMAPTNPSR1MEN1
SCHEMBL7613879 0.78 ALDH1A1 (0.56) ALDH1A1MAPTATMNPSR1MEN1
SCHEMBL9448980 0.77 CES2 (0.52) ALDH1A1LMNAMAPTNPSR1MEN1
SCHEMBL9448877 0.77 GPR52 (0.45) ALDH1A1LMNANPSR1MEN1KMT2A
SCHEMBL29883889 0.77 GPR52 (0.45) ALDH1A1LMNANPSR1MEN1KMT2A
SCHEMBL9449288 0.77 CES2 (0.52) ALDH1A1NPSR1MEN1KMT2AHTT
SCHEMBL6787746 0.76 NPSR1 (0.44) ALDH1A1LMNAMAPTATMNPSR1
SCHEMBL27201517 0.75 ALDH1A1 (0.51) ALDH1A1LMNATP53HSP90AA1MAPT
SCHEMBL15524099 0.75 ALDH1A1 (0.40) ALDH1A1TP53MAPTMEN1KMT2A
SCHEMBL8978021 0.74 NR4A1 (0.53) ALDH1A1LMNATP53MAPTNPSR1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0466730-B1 GEMINAL BISPHOSPHONIC ACIDS AND DERIVATIVES AS ANTI-ARTHRITIC AGENTS THE UPJOHN COMPANY (US) 1993-07-21 EP disclosed
US-5220021-A Geminal bisphosphonic acids and derivatives as anti-arthritic agents THE UPJOHN COMPANY (US) 1993-06-15 US disclosed
EP-0466730-A1 GEMINAL BISPHOSPHONIC ACIDS AND DERIVATIVES AS ANTI-ARTHRITIC AGENTS. UPJOHN CO (US) 1992-01-22 EP disclosed
WO-1990012017-A1 GEMINAL BISPHOSPHONIC ACIDS AND DERIVATIVES AS ANTI-ARTHRITIC AGENTS THE UPJOHN COMPANY (US) 1990-10-18 WO disclosed