SCHEMBL9449288

SCHEMBL9449288

[N-]=[N+]=CC(=O)c1ccccc1Cl

nearest known ligand 0.52

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CES2 O00748 1/20 0.52
CES1 P23141 1/20 0.52
ALDH1A1 P00352 2/20 0.50
POLB P06746 2/20 0.47
PTGS1 P23219 1/20 0.44
PTGS2 P35354 1/20 0.44
CYP1A2 P05177 2/20 0.42
HPGD P15428 2/20 0.42
CYP2C19 P33261 1/20 0.42
NPSR1 Q6W5P4 1/20 0.42
MEN1 O00255 1/20 0.41
HTT P42858 1/20 0.41
KMT2A Q03164 1/20 0.41
HIF1A Q16665 1/20 0.41
ERCC5 P28715 1/20 0.41
FEN1 P39748 1/20 0.41
RAB9A P51151 1/20 0.40
RECQL P46063 1/20 0.39
CXCL12 P48061 1/20 0.38
TSHR P16473 1/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9661974 0.86 ALDH1A1 (0.45) CES2CES1ALDH1A1POLBPTGS1
SCHEMBL9449000 0.78 ALDH1A1 (0.48) CES2CES1ALDH1A1CYP1A2HPGD
SCHEMBL7613879 0.78 ALDH1A1 (0.56) ALDH1A1POLBCYP1A2HPGDCYP2C19
SCHEMBL9449016 0.78 SMN1; SMN2 (0.53) ALDH1A1POLBHPGDMEN1HTT
SCHEMBL9448980 0.77 CES2 (0.52) CES2CES1ALDH1A1HPGDNPSR1
SCHEMBL9448951 0.77 ALDH1A1 (0.46) ALDH1A1POLBCYP1A2HPGDCYP2C19
SCHEMBL29883889 0.77 GPR52 (0.45) ALDH1A1HPGDNPSR1MEN1HTT
SCHEMBL9448877 0.77 GPR52 (0.45) ALDH1A1HPGDNPSR1MEN1HTT
SCHEMBL6787746 0.76 NPSR1 (0.44) ALDH1A1CYP1A2HPGDCYP2C19NPSR1
SCHEMBL9449241 0.76 ALDH1A1 (0.40) ALDH1A1NPSR1MEN1HTTKMT2A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0466730-B1 GEMINAL BISPHOSPHONIC ACIDS AND DERIVATIVES AS ANTI-ARTHRITIC AGENTS THE UPJOHN COMPANY (US) 1993-07-21 EP disclosed
US-5220021-A Geminal bisphosphonic acids and derivatives as anti-arthritic agents THE UPJOHN COMPANY (US) 1993-06-15 US disclosed
WO-1990012017-A1 GEMINAL BISPHOSPHONIC ACIDS AND DERIVATIVES AS ANTI-ARTHRITIC AGENTS THE UPJOHN COMPANY (US) 1990-10-18 WO disclosed