SCHEMBL9448980

SCHEMBL9448980

[N-]=[N+]=CC(=O)c1ccccc1F

nearest known ligand 0.52

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CES2 O00748 3/20 0.52
CES1 P23141 3/20 0.52
ALDH1A1 P00352 4/20 0.48
ALOX15 P16050 1/20 0.48
GPR52 Q9Y2T5 1/20 0.45
GAA P10253 1/20 0.44
MAOB P27338 1/20 0.44
MEN1 O00255 3/20 0.43
KMT2A Q03164 3/20 0.43
TDP1 Q9NUW8 1/20 0.43
MAPT P10636 2/20 0.42
NPSR1 Q6W5P4 2/20 0.42
NPC1 O15118 1/20 0.42
HPGD P15428 1/20 0.42
PTPN1 P18031 1/20 0.41
ERCC5 P28715 1/20 0.41
FEN1 P39748 1/20 0.41
HTT P42858 1/20 0.41
HIF1A Q16665 1/20 0.41
TSHR P16473 1/20 0.40

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8720874 0.85 CES2 (0.55) CES2CES1ALDH1A1ALOX15GAA
SCHEMBL7613879 0.78 ALDH1A1 (0.56) ALDH1A1ALOX15MEN1KMT2AMAPT
SCHEMBL295344 0.77 CES2 (0.62) CES2CES1ALDH1A1ALOX15GPR52
SCHEMBL9448951 0.77 ALDH1A1 (0.46) ALDH1A1MAOBMEN1KMT2AMAPT
SCHEMBL9449288 0.77 CES2 (0.52) CES2CES1ALDH1A1MEN1KMT2A
SCHEMBL29883889 0.77 GPR52 (0.45) ALDH1A1GPR52MEN1KMT2ANPSR1
SCHEMBL9448877 0.77 GPR52 (0.45) ALDH1A1GPR52MEN1KMT2ANPSR1
SCHEMBL6787746 0.76 NPSR1 (0.44) ALDH1A1MEN1KMT2AMAPTNPSR1
Water SCHEMBL29955657 0.75 CES2 (0.60) CES2CES1ALDH1A1ALOX15GPR52
Water SCHEMBL9329581 0.75 CES2 (0.60) CES2CES1ALDH1A1ALOX15GPR52

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0466730-B1 GEMINAL BISPHOSPHONIC ACIDS AND DERIVATIVES AS ANTI-ARTHRITIC AGENTS THE UPJOHN COMPANY (US) 1993-07-21 EP disclosed
US-5220021-A Geminal bisphosphonic acids and derivatives as anti-arthritic agents THE UPJOHN COMPANY (US) 1993-06-15 US disclosed
WO-1990012017-A1 GEMINAL BISPHOSPHONIC ACIDS AND DERIVATIVES AS ANTI-ARTHRITIC AGENTS THE UPJOHN COMPANY (US) 1990-10-18 WO disclosed